SCHEMBL21370171

SCHEMBL21370171

Cc1cc2ncnc(NC3CCCCC3)c2cc1C

nearest known ligand 0.71

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 5/20 0.71
TP53 P04637 1/20 0.53
USP2 O75604 1/20 0.52
LMNA P02545 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
TSHR P16473 1/20 0.52
CYP2C19 P33261 1/20 0.52
CLK4 Q9HAZ1 1/20 0.52
CD38 P28907 2/20 0.52
HPGDS O60760 1/20 0.50
EGFR P00533 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21369343 0.89 IRAK4 (0.65) IRAK4TP53USP2LMNACYP1A2
SCHEMBL17656914 0.87 IRAK4 (0.73) IRAK4USP2LMNACYP1A2CYP3A4
SCHEMBL19283376 0.83 IRAK4 (1.00) IRAK4
SCHEMBL19283377 0.83 IRAK4 (1.00) IRAK4
SCHEMBL17656917 0.82 IRAK4 (0.76) IRAK4
SCHEMBL7714365 0.81 IRAK4 (0.73) IRAK4USP2LMNACYP1A2CYP3A4
SCHEMBL29157226 0.78 IRAK4 (0.63) IRAK4CD38HPGDSEGFR
SCHEMBL6363833 0.78 CD38 (0.54) IRAK4TP53CD38HPGDSEGFR
SCHEMBL4357479 0.78 IRAK4 (0.75) IRAK4USP2LMNACYP1A2CYP3A4
SCHEMBL6367334 0.78 CD38 (0.54) IRAK4TP53CD38HPGDSEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3200788-B1 INHIBITORS OF IRAK4 ACTIVITY MERCK SHARP & DOHME (US) 2019-09-18 EP disclosed