SCHEMBL21372289

SCHEMBL21372289

O=c1ccc2ccc(=O)n3c2n1CC3CN1CCOC(CNCc2cc3c(cc2F)OCCO3)C1

nearest known ligand 0.38

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 1/20 0.37
KCNH2 Q12809 2/20 0.34
PKM P14618 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3328853 1.00 TOP2A (0.37) TOP2AKCNH2PKMKMT2A
Hydrochloric Acid SCHEMBL3367140 0.99 TOP2A (0.36) TOP2AKCNH2PKMKMT2A
SCHEMBL3364173 0.77 TOP2A (0.43) TOP2AKCNH2
SCHEMBL21372223 0.77 TOP2A (0.43) TOP2AKCNH2
Hydrochloric Acid SCHEMBL3367115 0.76 TOP2A (0.42) TOP2AKCNH2
SCHEMBL21372413 0.75 KCNH2 (0.38) TOP2AKCNH2
SCHEMBL3332295 0.75 KCNH2 (0.38) TOP2AKCNH2
Hydrochloric Acid SCHEMBL3333195 0.75 KCNH2 (0.37) TOP2AKCNH2
Hydrochloric Acid SCHEMBL3324139 0.75 TOP2A (0.33) TOP2A
SCHEMBL13299233 0.72 TOP2A (0.49) TOP2AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3639824-A1 TRICYCLIC NITROGEN CONTAINING COMPOUNDS FOR TREATING NEISSERIA GONORRHOEA INFECTION GlaxoSmithKline Intellectual Property Development Limited (GB) 2020-04-22 EP disclosed
EP-3182973-B1 TRICYCLIC NITROGEN CONTAINING COMPOUNDS FOR TREATING NEISSERIA GONORRHOEA INFECTION GLAXOSMITHKLINE IP DEV LTD (GB) 2019-09-18 EP disclosed