SCHEMBL21381373

SCHEMBL21381373

CCOC(=O)C(CC)C1CCN(C(=O)c2ccnc3ccc(F)cc23)CC1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GFER P55789 1/20 0.47
IDO1 P14902 5/20 0.46
KDM4E B2RXH2 1/20 0.44
HSD17B10 Q99714 1/20 0.44
ALDH1A1 P00352 6/20 0.43
MAPT P10636 2/20 0.42
TP53 P04637 1/20 0.42
POLB P06746 1/20 0.42
PREP P48147 1/20 0.42
SLC22A12 Q96S37 1/20 0.41
CYP2C19 P33261 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21385177 0.89 GFER (0.48) GFERIDO1KDM4EHSD17B10ALDH1A1
SCHEMBL21381380 0.89 IDO1 (0.52) GFERIDO1KDM4EHSD17B10ALDH1A1
SCHEMBL17729120 0.84 CHRM4 (0.54) IDO1MAPTTP53POLB
SCHEMBL21400820 0.81 IDO1 (0.59) GFERIDO1
SCHEMBL17729117 0.81 IDO1 (0.56) IDO1CYP2C19
SCHEMBL21400743 0.81 IDO1 (0.49) GFERIDO1KDM4EHSD17B10ALDH1A1
SCHEMBL21400827 0.79 IDO1 (0.56) GFERIDO1
SCHEMBL21400821 0.79 IDO1 (0.56) GFERIDO1
SCHEMBL21400826 0.79 IDO1 (0.56) GFERIDO1
SCHEMBL28699360 0.74 IDO1 (0.55) IDO1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111630043-B Compound containing ring, preparation method and application thereof in medicine 四川科伦博泰生物医药股份有限公司 2022-02-15 CN disclosed
CN-111630043-A Compound containing ring, preparation method and application thereof in medicine 四川科伦博泰生物医药股份有限公司 2020-09-04 CN disclosed
WO-2019179369-A1 RING-CONTAINING COMPOUND, PREPARATION METHOD THEREFOR, AND MEDICAL APPLICATION THEREOF 四川科伦博泰生物医药股份有限公司 2019-09-26 WO disclosed
WO-2019179369-A1 RING-CONTAINING COMPOUND, PREPARATION METHOD THEREFOR, AND MEDICAL APPLICATION THEREOF 四川科伦博泰生物医药股份有限公司 2019-09-26 WO disclosed