SCHEMBL2144015

SCHEMBL2144015

O=C(NO)c1cnc(N2CC3CC2CN3C(=O)C(c2ccccc2)c2ccccc2)nc1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 13/20 0.46
HDAC1 Q13547 13/20 0.46
HDAC2 Q92769 13/20 0.46
HDAC6 Q9UBN7 13/20 0.46
HDAC4 P56524 8/20 0.46
HDAC7 Q8WUI4 8/20 0.46
HDAC10 Q969S8 8/20 0.46
HDAC11 Q96DB2 8/20 0.46
HDAC8 Q9BY41 8/20 0.46
HDAC9 Q9UKV0 8/20 0.46
HDAC5 Q9UQL6 8/20 0.46
CHRNA7 P36544 1/20 0.42
KCNH2 Q12809 1/20 0.42
AGTR2 P50052 5/20 0.41
KDM1A O60341 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1365725 1.00 HDAC3 (0.46) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL1366758 0.84 HDAC6 (0.52) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL1366117 0.83 HDAC1 (0.45) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL1365029 0.83 HDAC6 (0.47) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL16302088 0.83 HDAC6 (0.47) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL1366934 0.82 HDAC1 (0.53) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL12142364 0.82 HDAC1 (0.53) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL2144014 0.78 HDAC1 (0.60) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL5062540 0.78 HDAC1 (0.60) HDAC3HDAC1HDAC2HDAC6HDAC4
SCHEMBL1364891 0.77 KCNH2 (0.49) HDAC3HDAC1HDAC2HDAC6HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2343286-A1 Dibenzo[b,f][1,4]oxazepine derivatives as inhibitors of histone deacetylase Methylgene, Inc. (CA) 2011-07-13 EP disclosed