SCHEMBL21442276

SCHEMBL21442276

C#CCOc1cnc(C(=O)Nc2ccc(F)c([C@H](C)CCOC(=N)N)c2)cn1

nearest known ligand 0.53

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.53
BACE2 Q9Y5Z0 6/20 0.52
CTSD P07339 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16006914 0.84 BACE1 (0.44) BACE1BACE2
SCHEMBL21442412 0.82 BACE1 (0.48) BACE1BACE2CTSD
SCHEMBL21442285 0.77 BACE1 (0.53) BACE1BACE2
SCHEMBL21442346 0.77 BACE1 (0.46) BACE1BACE2
SCHEMBL12445581 0.77 BACE1 (0.56) BACE1BACE2CTSD
SCHEMBL21442377 0.76 BACE1 (0.40) BACE1BACE2CTSD
SCHEMBL16006876 0.76 BACE1 (0.44) BACE1BACE2CTSD
SCHEMBL21442415 0.74 BACE1 (0.49) BACE1BACE2CTSD
SCHEMBL21442374 0.74 BACE1 (0.40) BACE1BACE2
SCHEMBL20852120 0.73 NPC1 (0.56) BACE1BACE2CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2961749-B1 PERFLUORINATED 5,6-DIHYDRO-4H-1,3-OXAZIN-2-AMINE COMPOUNDS AS BETA-SECRETASE INHIBITORS AND METHODS OF USE AMGEN INC (US) 2019-10-09 EP disclosed