SCHEMBL21443514

SCHEMBL21443514

CCC(=O)Nc1cccc(Oc2nc(Nc3cccc(N4CCN(CCO)CC4)c3)ncc2F)c1

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EGFR P00533 18/20 0.60
NUAK2 Q9H093 2/20 0.56
NUAK1 O60285 1/20 0.56
ITK Q08881 4/20 0.51
JAK2 O60674 1/20 0.48
BLK P51451 1/20 0.48
BMX P51813 1/20 0.48
JAK3 P52333 1/20 0.48
BTK Q06187 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2228637 0.89 EGFR (0.78) EGFRNUAK2NUAK1ITKJAK2
SCHEMBL29722352 0.89 EGFR (0.78) EGFRNUAK2NUAK1ITKJAK2
SCHEMBL13166469 0.79 EGFR (0.80) EGFRNUAK2NUAK1ITKBTK
SCHEMBL16391084 0.76 EGFR (0.69) EGFRNUAK1ITKJAK2BLK
SCHEMBL29722245 0.75 EGFR (1.00) EGFRITKJAK3BTK
SCHEMBL13165553 0.75 EGFR (1.00) EGFRITKJAK3BTK
SCHEMBL18165638 0.75 EGFR (0.65) EGFRITKJAK2BLKBMX
SCHEMBL23450611 0.74 BTK (0.71) EGFRJAK2BLKJAK3BTK
SCHEMBL16391080 0.74 EGFR (0.65) EGFRITKJAK2BLKBMX
SCHEMBL31060495 0.72 EGFR (1.00) EGFRNUAK2NUAK1ITKJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3549934-A1 HETEROARYL COMPOUNDS AND USES THEREOF Celgene CAR LLC (BM) 2019-10-09 EP disclosed