SCHEMBL21451973

SCHEMBL21451973

Cc1nc2c(s1)CN(CCCN1CCOCC1)CC2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.49
GRM5 P41594 3/20 0.43
RAD52 P43351 1/20 0.43
RECQL P46063 1/20 0.43
DRD2 P14416 2/20 0.37
DRD3 P35462 2/20 0.37
PDE10A Q9Y233 2/20 0.36
KEAP1 Q14145 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HDAC6 Q9UBN7 1/20 0.35
HTR2A P28223 1/20 0.35
MYC P01106 1/20 0.35
KDM1A O60341 1/20 0.35
TNNI3K Q59H18 1/20 0.35
KDM4E B2RXH2 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
PKM P14618 1/20 0.34
APOBEC3G Q9HC16 1/20 0.34
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14907151 0.89 HRH3 (0.49) HRH3DRD2DRD3KEAP1SMN1; SMN2
SCHEMBL14907159 0.86 HRH3 (0.46) HRH3DRD2DRD3KEAP1SMN1; SMN2
SCHEMBL17383827 0.81 RAD52 (0.48) HRH3GRM5RAD52RECQLDRD2
SCHEMBL12680942 0.80 RAD52 (0.53) HRH3GRM5RAD52RECQLDRD2
SCHEMBL16286091 0.79 RAD52 (0.48) HRH3GRM5RAD52RECQLDRD2
SCHEMBL21451980 0.78 HRH3 (0.43) HRH3GRM5RAD52RECQLPDE10A
SCHEMBL21451967 0.77 GRM5 (0.45) HRH3GRM5RAD52RECQLSMN1; SMN2
SCHEMBL21451976 0.76 HRH3 (0.47) HRH3GRM5RAD52RECQLDRD2
SCHEMBL12344273 0.76 HRH3 (0.47) HRH3GRM5RAD52RECQLDRD2
SCHEMBL6369558 0.76 RAD52 (0.69) HRH3GRM5RAD52RECQLPDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019192506-A1 IMMUNOMODULATORS, COMPOSITIONS AND METHODS THEREOF BETTA PHARMACEUTICALS CO., LTD (CN) 2019-10-10 WO disclosed