SCHEMBL21452563

SCHEMBL21452563

O=NC1(c2cccc(OC(F)(F)F)c2F)CCCCC1=O

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MPL P40238 1/20 0.33
GRIA1 P42261 1/20 0.32
CACNG8 Q8WXS5 1/20 0.32
GRIN1 Q05586 3/20 0.32
GRIN2A Q12879 3/20 0.32
GRIN2D O15399 2/20 0.32
GRIN3B O60391 2/20 0.32
GRIN2B Q13224 2/20 0.32
GRIN2C Q14957 2/20 0.32
GRIN3A Q8TCU5 2/20 0.32
SLC6A9 P48067 1/20 0.32
DDB1 Q16531 2/20 0.31
CRBN Q96SW2 2/20 0.31
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
HDAC4 P56524 1/20 0.31
SLC6A4 P31645 2/20 0.30
OPRK1 P41145 1/20 0.30
LMNA P02545 1/20 0.30
OPRM1 P35372 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21452512 0.81 PDE7A (0.40) MPLGRIN1GRIN2AGRIN2DGRIN3B
SCHEMBL21451904 0.80 HDAC4 (0.48) GRIN1GRIN2AGRIN2DGRIN3BGRIN2B
SCHEMBL21451925 0.80 MPL (0.37) MPLGRIA1CACNG8GRIN1GRIN2A
SCHEMBL21452196 0.80 MPL (0.37) MPLGRIA1CACNG8GRIN1GRIN2A
SCHEMBL21452197 0.80 MPL (0.37) MPLGRIA1CACNG8GRIN1GRIN2A
SCHEMBL21452460 0.78 GRIN1 (0.45) GRIN1GRIN2AGRIN2DGRIN3BGRIN2B
SCHEMBL23490936 0.76 MPL (0.32) MPLGRIN1GRIN2AGRIN2DGRIN3B
SCHEMBL21451922 0.76 HCRTR1 (0.34) GRIN1GRIN2AGRIN2BHCRTR1HCRTR2
SCHEMBL25381960 0.75 HDAC4 (0.36) GRIN1GRIN2AGRIN2DGRIN3BGRIN2B
SCHEMBL29077176 0.74 HDAC4 (0.33) MPLGRIN1GRIN2AGRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3778579-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Jianhe Pharmaceutical & Technology Co. Ltd. (CN) 2021-02-17 EP disclosed
WO-2019192602-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海键合医药科技有限公司 2019-10-10 WO disclosed