SCHEMBL21456776

SCHEMBL21456776

CC(=O)N1CCC(CCC(=O)Nc2cc(-c3cccs3)ccc2[AsH2])CC1

nearest known ligand 0.67

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 20/20 0.67
HDAC2 Q92769 20/20 0.67
HDAC3 O15379 16/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13833516 0.89 HDAC1 (0.84) HDAC1HDAC2HDAC3
SCHEMBL13736302 0.80 HDAC1 (1.00) HDAC1HDAC2HDAC3
SCHEMBL13833485 0.80 HDAC1 (0.79) HDAC1HDAC2HDAC3
SCHEMBL13735538 0.76 HDAC1 (1.00) HDAC1HDAC2HDAC3
SCHEMBL13739871 0.74 HDAC1 (0.79) HDAC1HDAC2HDAC3
SCHEMBL13833455 0.74 HDAC1 (1.00) HDAC1HDAC2HDAC3
SCHEMBL13735278 0.73 HDAC1 (0.74) HDAC1HDAC2HDAC3
SCHEMBL13833318 0.73 HDAC2 (1.00) HDAC1HDAC2HDAC3
SCHEMBL13833334 0.73 HDAC2 (1.00) HDAC1HDAC2HDAC3
SCHEMBL13736754 0.72 HDAC1 (0.53) HDAC1HDAC2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2701699-B1 INHIBITORS OF HISTONE DEACETYLASE BROAD INST INC (US) 2019-10-16 EP disclosed