SCHEMBL21494470

SCHEMBL21494470

CCOc1cc(C(CC(=O)OC)N2C(=O)c3cccc([N+](=O)[O-])c3C2=O)ccc1OC.O=C1OC(=O)c2c1cccc2[N+](=O)[O-]

nearest known ligand 0.79

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TNF P01375 8/20 0.79
PDE4A P27815 13/20 0.66
PDE4B Q07343 13/20 0.66
PDE4C Q08493 13/20 0.66
PDE4D Q08499 13/20 0.66
HTR2B P41595 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30568370 0.94 TNF (0.88) TNFPDE4APDE4BPDE4CPDE4D
SCHEMBL7741608 0.94 TNF (0.88) TNFPDE4APDE4BPDE4CPDE4D
SCHEMBL30568371 0.94 TNF (0.88) TNFPDE4APDE4BPDE4CPDE4D
SCHEMBL23000632 0.87 TNF (0.75) TNFPDE4APDE4BPDE4CPDE4D
SCHEMBL6098123 0.87 TNF (0.75) TNFPDE4APDE4BPDE4CPDE4D
SCHEMBL23000615 0.87 TNF (0.75) TNFPDE4APDE4BPDE4CPDE4D
SCHEMBL825659 0.86 TNF (0.74) TNFPDE4APDE4BPDE4CPDE4D
SCHEMBL7433881 0.83 TNF (0.68) TNFPDE4APDE4BPDE4CPDE4D
SCHEMBL21494496 0.82 TNF (0.87) TNFPDE4APDE4BPDE4CPDE4D
SCHEMBL21494520 0.82 TNF (0.87) TNFPDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019201255-A1 ISOINDOLE DERIVATIVE 天津合美医药科技有限公司 2019-10-24 WO disclosed