SCHEMBL21494876

SCHEMBL21494876

COc1cc(=O)[nH]c(C)n1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.48
HPGD P15428 1/20 0.46
TSHR P16473 1/20 0.46
CASP7 P55210 1/20 0.46
GSK3B P49841 1/20 0.44
KDM4E B2RXH2 3/20 0.41
LMNA P02545 2/20 0.41
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 1/20 0.39
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
ALDH1A1 P00352 1/20 0.38
PDE2A O00408 1/20 0.38
CYP19A1 P11511 2/20 0.38
NQO2 P16083 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26980532 0.78 CYP3A4 (0.55) HPGDTSHRCASP7KDM4EMEN1
SCHEMBL2632907 0.74
SCHEMBL5935763 0.73
SCHEMBL7161983 0.70
SCHEMBL11937375 0.70
SCHEMBL18689667 0.70
SCHEMBL13375700 0.70
SCHEMBL26910344 0.69 PDE2A (0.50) PDE2A
SCHEMBL18643546 0.69 TYMS (0.43) HPGDKDM4ELMNAHSD17B10PDE3B
SCHEMBL10684112 0.68 ADORA2A (0.61) HPGDTSHRGSK3BKDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3781565-A1 2-METHYL-AZA-QUINAZOLINES Bayer Pharma Aktiengesellschaft (DE) 2021-02-24 EP disclosed
WO-2019201848-A1 2-METHYL-AZA-QUINAZOLINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2019-10-24 WO disclosed