SCHEMBL21496716

SCHEMBL21496716

CC1(C)c2cccc(C(N)=O)c2CN1C(=O)Nc1ccc(C(F)(F)F)nc1

nearest known ligand 0.81

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC11 Q96DB2 8/20 0.81
HDAC8 Q9BY41 1/20 0.51
TRPV1 Q8NER1 1/20 0.43
AR P10275 3/20 0.38
JAK2 O60674 4/20 0.37
JAK1 P23458 4/20 0.37
USP30 Q70CQ3 1/20 0.36
CDK5 Q00535 1/20 0.36
CDK5R1 Q15078 1/20 0.36
PTGES O14684 1/20 0.36
EPHX2 P34913 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21496663 0.90 HDAC11 (0.80) HDAC11HDAC8TRPV1ARUSP30
SCHEMBL21496846 0.90 HDAC11 (1.00) HDAC11HDAC8TRPV1ARUSP30
SCHEMBL21496665 0.85 HDAC11 (0.59) HDAC11HDAC8TRPV1EPHX2
SCHEMBL21496660 0.76 HDAC11 (0.79) HDAC11HDAC8
SCHEMBL30039900 0.76 HDAC11 (0.75) HDAC11HDAC8
SCHEMBL21500576 0.76 HDAC11 (0.75) HDAC11HDAC8
SCHEMBL25932218 0.75 HDAC11 (0.59) HDAC11HDAC8
SCHEMBL25932217 0.75 HDAC11 (0.76) HDAC11HDAC8
SCHEMBL21496849 0.74 HDAC11 (0.74) HDAC11HDAC8
SCHEMBL21496709 0.74 HDAC11 (0.58) HDAC11HDAC8TRPV1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3784654-A1 ISOINDOLINES AS HDAC INHIBITORS Valo Early Discovery, Inc. (US) 2021-03-03 EP disclosed
WO-2019204550-A1 ISOINDOLINES AS HDAC INHIBITORS FORMA THERAPEUTICS, INC. (US) 2019-10-24 WO disclosed