SCHEMBL21503

SCHEMBL21503

CS(=O)(=O)c1c(N)n2ncc(-c3cnn(-c4ccccc4)c3)c2nc1[C@H]1CC[C@@H](C(N)=O)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 17/20 0.41
CCNA2 P20248 16/20 0.41
CDK2 P24941 16/20 0.41
CCNA1 P78396 16/20 0.41
GRM2 Q14416 1/20 0.38
TYK2 P29597 1/20 0.38
PIM1 P11309 2/20 0.37
MAP2K2 P36507 2/20 0.37
NTRK1 P04629 1/20 0.37
MET P08581 1/20 0.37
FGFR1 P11362 1/20 0.37
FLT3 P36888 1/20 0.37
MAPK8 P45983 1/20 0.37
GSK3B P49841 1/20 0.37
NTRK3 Q16288 1/20 0.37
ALK Q9UM73 1/20 0.37
DYRK1B Q9Y463 1/20 0.37
RPS6KA4 O75676 1/20 0.36
STK10 O94804 1/20 0.36
LATS1 O95835 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26939 0.85 CHEK1 (0.41) CHEK1CCNA2CDK2CCNA1GRM2
Bicarbonate SCHEMBL17836378 0.84 CHEK1 (0.37) CHEK1CCNA2CDK2CCNA1GRM2
SCHEMBL15007376 0.82 CHEK1 (0.35) CHEK1CCNA2CDK2CCNA1GRM2
SCHEMBL15031503 0.82 CHEK1 (0.35) CHEK1CCNA2CDK2CCNA1GRM2
SCHEMBL15007377 0.82 CHEK1 (0.35) CHEK1CCNA2CDK2CCNA1GRM2
SCHEMBL31398 0.82 CHEK1 (0.33) CHEK1CCNA2CDK2CCNA1TYK2
SCHEMBL28745 0.81 CHEK1 (0.36) CHEK1CCNA2CDK2CCNA1GRM2
SCHEMBL28827 0.81 CHEK1 (0.36) CHEK1CCNA2CDK2CCNA1GRM2
SCHEMBL20975 0.81 CHEK1 (0.36) CHEK1CCNA2CDK2CCNA1GRM2
SCHEMBL10236906 0.80 CHEK1 (0.42) CHEK1CCNA2CDK2CCNA1GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012027236-A1 NOVEL PYRAZOLO[1,5-a]PYRIMIDINE DERIVATIVES AS mTOR INHIBITORS SCHERING CORPORATION (US) 2012-03-01 WO disclosed