SCHEMBL21538871

SCHEMBL21538871

C=CC(Cc1cccc(C(F)(F)F)c1)C(=C)C

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.55
HTR2B P41595 3/20 0.55
HTR2C P28335 2/20 0.55
SIGMAR1 Q99720 2/20 0.49
ADRA2C P18825 2/20 0.49
SLC6A4 P31645 2/20 0.49
ADRA1A P35348 2/20 0.49
DRD3 P35462 2/20 0.49
LMNA P02545 1/20 0.49
MAPT P10636 1/20 0.49
OPRK1 P41145 1/20 0.49
ACP3 P15309 1/20 0.43
CYP3A4 P08684 3/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2D6 P10635 2/20 0.43
TP53 P04637 1/20 0.43
TSHR P16473 1/20 0.43
CYP2C19 P33261 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43
EPHX1 P07099 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21076021 0.79 HTR2A (0.60) HTR2AHTR2BHTR2CSIGMAR1ADRA2C
SCHEMBL18739763 0.75 HTR2A (0.64) HTR2AHTR2BHTR2CSIGMAR1ADRA2C
SCHEMBL18739769 0.75 HTR2A (0.64) HTR2AHTR2BHTR2CSIGMAR1ADRA2C
SCHEMBL30412479 0.73 HTR2A (0.72) HTR2AHTR2BHTR2CSIGMAR1ADRA2C
SCHEMBL5706525 0.73 HTR2A (0.72) HTR2AHTR2BHTR2CSIGMAR1ADRA2C
SCHEMBL5706540 0.73 HTR2A (0.72) HTR2AHTR2BHTR2CSIGMAR1ADRA2C
SCHEMBL21306789 0.73 HTR2A (0.53) HTR2AHTR2BHTR2CSIGMAR1ADRA2C
SCHEMBL2421761 0.73 HTR2A (0.72) HTR2AHTR2BHTR2CSIGMAR1ADRA2C
SCHEMBL28256765 0.73 HTR2A (0.72) HTR2AHTR2BHTR2CSIGMAR1ADRA2C
SCHEMBL19040919 0.73 HTR2A (0.71) HTR2AHTR2BHTR2CSIGMAR1ADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3560920-A1 SECONDARY ALCOHOL QUINOLINYL MODULATORS OF ROR GAMMA T Janssen Pharmaceutica NV (BE) 2019-10-30 EP disclosed