SCHEMBL21554467

SCHEMBL21554467

Clc1cnc(OC2CCOC2)nc1-n1cnc2ccccc21

nearest known ligand 0.67

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
MKNK2 Q9HBH9 15/20 0.67
MKNK1 Q9BUB5 18/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21554266 0.94 MKNK2 (0.76) MKNK2MKNK1
SCHEMBL21554334 0.94 MKNK1 (0.66) MKNK2MKNK1
SCHEMBL21554301 0.86 MKNK2 (0.89) MKNK2MKNK1
SCHEMBL21554270 0.85 MKNK1 (0.70) MKNK2MKNK1
SCHEMBL21554281 0.81 MKNK1 (0.74) MKNK2MKNK1
SCHEMBL22722390 0.81 MKNK1 (0.74) MKNK2MKNK1
SCHEMBL20479143 0.81 MKNK1 (0.74) MKNK2MKNK1
SCHEMBL22722382 0.81 MKNK1 (0.74) MKNK2MKNK1
SCHEMBL21554508 0.81 MKNK1 (0.64) MKNK2MKNK1
SCHEMBL21554336 0.81 MKNK1 (0.64) MKNK2MKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10851082-B2 Substituted aromatic n-heterocyclic compounds as inhibitors of mitogen-activated protein kinase interacting kinase 1 (MNK1) and 2 (MNK2) NORTHWESTERN UNIVERSITY (US) 2020-12-01 US disclosed
EP-3564235-A1 SUBSTITUTED AROMATIC N-HETEROCYCLIC COMPOUNDS AS INHIBITORS OF MITOGEN-ACTIVATED PROTEIN KINASE INTERACTING KINASE 1 (MNK1) AND 2 (MNK2) Northwestern University (US) 2019-11-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10851082-B2 Substituted aromatic n-heterocyclic compounds as inhibitors of mitogen-activated protein kinase interacting kinase 1 (MNK1) and 2 (MNK2) MAP4K2, MAP3K20, MKNK2 MKNK2 3/4885MKNK1 5/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.