SCHEMBL21556645

SCHEMBL21556645

CS(=O)(=O)N1CC[C@@H](NI)C1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.42
ALDH1A1 P00352 2/20 0.41
TSHR P16473 3/20 0.39
EPHX2 P34913 3/20 0.39
KDM1A O60341 1/20 0.39
EPHX1 P07099 1/20 0.39
FABP6 P51161 1/20 0.38
LMNA P02545 1/20 0.37
NPSR1 Q6W5P4 1/20 0.35
SMYD3 Q9H7B4 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
MAPK1 P28482 1/20 0.34
MAPT P10636 1/20 0.34
IDO1 P14902 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12820441 1.00 TP53 (0.42) TP53ALDH1A1TSHREPHX2KDM1A
SCHEMBL12820051 0.88 TP53 (0.48) TP53ALDH1A1TSHREPHX2KDM1A
SCHEMBL765729 0.82 TP53 (0.43) TP53ALDH1A1TSHREPHX2KDM1A
SCHEMBL962299 0.82 TP53 (0.43) TP53ALDH1A1TSHREPHX2KDM1A
SCHEMBL12225575 0.82 TP53 (0.43) TP53ALDH1A1TSHREPHX2KDM1A
SCHEMBL962569 0.82 TP53 (0.43) TP53ALDH1A1TSHREPHX2KDM1A
SCHEMBL26309055 0.78 TP53 (0.41) TP53ALDH1A1TSHREPHX2KDM1A
SCHEMBL12404074 0.78 TP53 (0.41) TP53ALDH1A1TSHREPHX2KDM1A
SCHEMBL12404082 0.78 TP53 (0.41) TP53ALDH1A1TSHREPHX2KDM1A
SCHEMBL12750460 0.77 FABP6 (0.42) TP53ALDH1A1TSHREPHX2KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3221306-B1 HETEROARYL COMPOUNDS AS IRAK INHIBITORS AND USES THEREOF MERCK PATENT GMBH (DE) 2019-11-13 EP disclosed