SCHEMBL21580368

SCHEMBL21580368

CC(C)(C)OC(=O)/N=C(/NC(=O)OC(C)(C)C)NC1CC(C(=O)O)C1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.49
NFKB1 P19838 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
KMT2A Q03164 3/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
GAA P10253 2/20 0.33
KDM1A O60341 1/20 0.33
MAOB P27338 1/20 0.33
EPHX1 P07099 1/20 0.33
CTSK P43235 2/20 0.32
MEN1 O00255 1/20 0.31
MAPK1 P28482 1/20 0.31
EPHX2 P34913 1/20 0.30
CYP2C9 P11712 1/20 0.30
HSD11B1 P28845 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9611663 0.84 BTK (0.35) BTKNFKB1NFKB2RELAKMT2A
SCHEMBL15489159 0.84 BTK (0.35) BTKNFKB1NFKB2RELAKMT2A
SCHEMBL13892845 0.82 BTK (0.38) BTKNFKB1NFKB2RELAKDM1A
SCHEMBL15632420 0.82 BTK (0.39) BTKKMT2AL3MBTL1CTSKMEN1
SCHEMBL19508986 0.81 GAA (0.39) BTKNFKB1NFKB2RELAKMT2A
SCHEMBL18256753 0.81 GAA (0.39) BTKNFKB1NFKB2RELAKMT2A
SCHEMBL10108121 0.80 BTK (0.35) BTKNFKB1NFKB2RELAKMT2A
SCHEMBL10108126 0.80 BTK (0.35) BTKNFKB1NFKB2RELAKMT2A
SCHEMBL10329511 0.80 BTK (0.47) BTKKMT2AL3MBTL1GAAKDM1A
SCHEMBL22233303 0.80 EPHX1 (0.40) BTKNFKB1NFKB2RELAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE47741-E1 Antibacterial aminoglycoside analogs ACHAOGEN, INC. (US) 2019-11-26 US disclosed