SCHEMBL21585963

SCHEMBL21585963

CCCCC1(CCCC)CN(c2ccc(OC)cc2)c2cc(SC)c(OC=C(F)C(=O)O)cc2S(O)(O)C1

nearest known ligand 0.36

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.36
SLC10A2 Q12908 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22476251 1.00 NR1H4 (0.36) NR1H4SLC10A2
SCHEMBL28530679 0.93 NR1H4 (0.37) NR1H4SLC10A2
SCHEMBL21585960 0.93 NR1H4 (0.37) NR1H4SLC10A2
SCHEMBL21585999 0.92 NR1H4 (0.40) NR1H4
SCHEMBL22476235 0.92 NR1H4 (0.40) NR1H4
SCHEMBL23451427 0.92 NR1H4 (0.35) NR1H4SLC10A2
SCHEMBL22476264 0.92 NR1H4 (0.35) NR1H4
SCHEMBL21585954 0.92 NR1H4 (0.40) NR1H4
SCHEMBL21585956 0.92 NR1H4 (0.40) NR1H4
SCHEMBL29189012 0.92 NR1H4 (0.34) NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3802504-A1 BENZOTHIA(DI)AZEPINE COMPOUNDS AND THEIR USE AS BILE ACID MODULATORS Albireo AB (SE) 2021-04-14 EP disclosed
CN-112449637-A Benzothia (di) azepanes and their use as bile acid modulators 阿尔比里奥公司 2021-03-05 CN disclosed
WO-2019234077-A1 BENZOTHIA(DI)AZEPINE COMPOUNDS AND THEIR USE AS BILE ACID MODULATORS ALBIREO AB (SE) 2019-12-12 WO disclosed