SCHEMBL21595660

SCHEMBL21595660

OCCOc1ccc(Cl)cc1F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR4 O95977 3/20 0.48
MRGPRX4 Q96LA9 1/20 0.48
PTGS2 P35354 2/20 0.45
PRKAB2 O43741 2/20 0.45
PRKAG1 P54619 2/20 0.45
PRKAA2 P54646 2/20 0.45
PRKAA1 Q13131 2/20 0.45
PRKAG3 Q9UGI9 2/20 0.45
PRKAG2 Q9UGJ0 2/20 0.45
PRKAB1 Q9Y478 2/20 0.45
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
PPARG P37231 6/20 0.43
PPARA Q07869 5/20 0.43
FFAR1 O14842 1/20 0.43
PPARD Q03181 1/20 0.43
HTR1A P08908 1/20 0.42
HTR7 P34969 1/20 0.42
TP53 P04637 1/20 0.41
MAPK1 P28482 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25218653 0.91 S1PR4 (0.47) S1PR4MRGPRX4PRKAB2PRKAG1PRKAA2
SCHEMBL21601495 0.83 S1PR4 (0.49) S1PR4MRGPRX4PPARGPPARAFFAR1
SCHEMBL30025714 0.81 S1PR4 (0.48) S1PR4MRGPRX4PPARGPPARAFFAR1
SCHEMBL5317553 0.81 S1PR4 (0.48) S1PR4MRGPRX4PPARGPPARAFFAR1
SCHEMBL19555362 0.81 S1PR4 (0.48) S1PR4MRGPRX4PPARGPPARAFFAR1
SCHEMBL3864712 0.81 ALOX5AP (0.44) PTGS2PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL4334537 0.81 S1PR4 (0.61) S1PR4MRGPRX4TP53MAPK1L3MBTL1
SCHEMBL5318910 0.80 S1PR4 (0.47) S1PR4MRGPRX4LMNAPPARGPPARA
SCHEMBL2252284 0.79 MRGPRX4 (0.48) S1PR4MRGPRX4PPARGPPARAFFAR1
SCHEMBL12505493 0.78 MAPT (0.49) S1PR4ALDH1A1LMNATP53MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019244066-A2 PYRIDIN-3-YL ACETIC ACID DERIVATIVES AS INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION VIIV Healthcare UK (No.5) Limited (GB) 2019-12-26 WO disclosed
WO-2019244066-A2 PYRIDIN-3-YL ACETIC ACID DERIVATIVES AS INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION VIIV Healthcare UK (No.5) Limited (GB) 2019-12-26 WO disclosed