SCHEMBL21595891

SCHEMBL21595891

NCCOc1ccc(F)cc1Cl

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.48
S1PR4 O95977 2/20 0.48
CSNK2A1 P68400 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.46
GLA P06280 1/20 0.46
DHFR P00374 2/20 0.46
RAB9A P51151 4/20 0.43
NPC1 O15118 3/20 0.43
SLC6A2 P23975 2/20 0.42
SLC6A3 Q01959 2/20 0.42
SLC6A4 P31645 1/20 0.42
PARP1 P09874 1/20 0.41
PARP3 Q9Y6F1 1/20 0.41
MAPT P10636 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
HTR1B P28222 1/20 0.41
HPGD P15428 1/20 0.41
ATM Q13315 1/20 0.41
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2252697 0.87 S1PR4 (0.49) S1PR4CSNK2A1DHFRRAB9ANPC1
SCHEMBL8959114 0.85 HTR2A (0.47) SMN1; SMN2GLASLC6A4
SCHEMBL8959084 0.84 PPARA (0.56) SMN1; SMN2GLA
SCHEMBL11669016 0.83 S1PR4 (0.49) S1PR4CSNK2A1SMN1; SMN2DHFRRAB9A
SCHEMBL29546953 0.82 KDM4E (0.54) KDM4EDHFRRAB9APARP1PARP3
SCHEMBL21601494 0.82 KDM4E (0.54) KDM4EDHFRRAB9APARP1PARP3
SCHEMBL10359829 0.81 S1PR4 (0.48) S1PR4DHFRRAB9ANPC1SLC6A2
SCHEMBL3453883 0.81 S1PR4 (0.54) S1PR4CSNK2A1RAB9ANPC1MAPT
Hydrochloric Acid SCHEMBL7425078 0.81 KDM4E (0.57) KDM4ESMN1; SMN2RAB9APARP1PARP3
SCHEMBL8959126 0.80 PPARA (0.48) SMN1; SMN2GLASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019244066-A2 PYRIDIN-3-YL ACETIC ACID DERIVATIVES AS INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION VIIV Healthcare UK (No.5) Limited (GB) 2019-12-26 WO disclosed
WO-2019244066-A2 PYRIDIN-3-YL ACETIC ACID DERIVATIVES AS INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION VIIV Healthcare UK (No.5) Limited (GB) 2019-12-26 WO disclosed