SCHEMBL21610175

SCHEMBL21610175

CC1(C)NC(=O)N(c2ccnc(Oc3ccc4c(c3)OC(F)(F)O4)n2)C1=O

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AR P10275 7/20 0.38
NOTUM Q6P988 1/20 0.34
ATP4A P20648 1/20 0.33
ATP4B P51164 1/20 0.33
NOS2 P35228 2/20 0.33
RXRA P19793 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2B Q13224 1/20 0.33
CYP1A2 P05177 1/20 0.33
MRGPRX4 Q96LA9 1/20 0.32
PDE2A O00408 2/20 0.32
KIT P10721 4/20 0.32
BRAF P15056 4/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21610193 0.83 AR (0.37) ARNOTUMMRGPRX4
SCHEMBL21580779 0.83 AR (0.37) ARNOTUMMRGPRX4
SCHEMBL21580766 0.81 AR (0.49) ARNOTUMRXRAGRIN1GRIN2B
SCHEMBL21610186 0.81 AR (0.37) ARMRGPRX4
SCHEMBL21610141 0.80 AR (0.40) AR
SCHEMBL21610232 0.78 AR (0.38) AR
SCHEMBL21610234 0.77 AR (0.37) AR
SCHEMBL21610266 0.76 AR (0.38) ARBRAF
SCHEMBL21610206 0.76 AR (0.43) ARCYP1A2MRGPRX4BRAF
SCHEMBL21610154 0.76 AR (0.41) ARCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220112176-A1 SUBSTITUTED-N-HETEROARYL COMPOUNDS AND USES THEREOF BIONOMICS LIMITED (AU) 2022-04-14 US disclosed
EP-3947365-A2 SUBSTITUTED-N-HETEROARYL COMPOUNDS AND USES THEREOF Bionomics Limited (AU) 2022-02-09 EP disclosed
WO-2020000065-A2 SUBSTITUTED-N-HETEROARYL COMPOUNDS AND USES THEREOF BIONOMICS LIMITED (AU) 2020-01-02 WO disclosed
WO-2020000065-A2 SUBSTITUTED-N-HETEROARYL COMPOUNDS AND USES THEREOF BIONOMICS LIMITED (AU) 2020-01-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220112176-A1 SUBSTITUTED-N-HETEROARYL COMPOUNDS AND USES THEREOF GABRE, GRIN2C, GRIN2A AR 4592/4885NOTUM 1160/4885ATP4A 2643/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.