SCHEMBL21658744

SCHEMBL21658744

Cc1nc2c(F)cc(-c3nc(Nc4ccc(CN5CCCC(C)C5)cn4)ncc3F)cc2n1C(C)C

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 20/20 0.76
CDK6 Q00534 15/20 0.76
CDK1 P06493 13/20 0.76
CCND3 P30281 12/20 0.76
CDK2 P24941 7/20 0.76
CCNE1 P24864 6/20 0.76
CCNA2 P20248 5/20 0.76
CCNB1 P14635 5/20 0.76
CDK9 P50750 4/20 0.76
CCNT1 O60563 3/20 0.76
CDK7 P50613 3/20 0.76
CCNH P51946 2/20 0.76
CIT O14578 1/20 0.76
GAK O14976 1/20 0.76
DYRK3 O43781 1/20 0.76
STK16 O75716 1/20 0.76
CCNK O75909 1/20 0.76
STK10 O94804 1/20 0.76
PRKD3 O94806 1/20 0.76
ABCB11 O95342 1/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17488913 0.92 CDK4 (0.75) CDK4CDK6CDK1CCND3CDK2
SCHEMBL17488639 0.92 CDK4 (0.75) CDK4CDK6CDK1CCND3CDK2
SCHEMBL17488760 0.91 CDK4 (0.88) CDK4CDK6CDK1CCND3CDK2
SCHEMBL21658739 0.90 CDK4 (0.87) CDK4CDK6CDK1CCND3CDK2
SCHEMBL17488747 0.89 CDK4 (0.77) CDK4CDK6CDK1CCND3CDK2
SCHEMBL30352281 0.89 CDK4 (0.84) CDK4CDK6CDK1CCND3CDK2
SCHEMBL17489209 0.88 CDK4 (0.76) CDK4CDK6CDK1CCND3CDK2
SCHEMBL17489053 0.88 CDK4 (0.76) CDK4CDK6CDK1CCND3CDK2
SCHEMBL17489278 0.88 CDK4 (0.76) CDK4CDK6CDK1CCND3CDK2
SCHEMBL17489244 0.88 CDK4 (0.76) CDK4CDK6CDK1CCND3CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020023917-A1 CDK INHIBITORS AND USES THEREOF CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2020-01-30 WO disclosed