SCHEMBL21669909

SCHEMBL21669909

CCOc1ccc(CC(NS(C)(=O)=O)C(=O)NC(Cc2ccccc2)C(=O)NCc2ccc(CNC(=O)OC(C)(C)C)cc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 19/20 0.61
KLK1 P06870 6/20 0.55
PSMB1 P20618 1/20 0.52
PSMB9 P28065 1/20 0.52
PSMB10 P40306 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14485476 1.00 KLKB1 (0.61) KLKB1KLK1PSMB1PSMB9PSMB10
SCHEMBL14485437 0.88 KLKB1 (0.64) KLKB1KLK1
SCHEMBL14485441 0.88 KLKB1 (0.64) KLKB1KLK1
SCHEMBL14485398 0.88 KLKB1 (0.70) KLKB1KLK1
SCHEMBL14485400 0.88 KLKB1 (0.70) KLKB1KLK1
SCHEMBL14554987 0.87 KLKB1 (0.79) KLKB1KLK1
Benzene SCHEMBL14486117 0.87 KLKB1 (0.79) KLKB1KLK1
SCHEMBL15901012 0.87 KLKB1 (0.61) KLKB1KLK1PSMB1PSMB9PSMB10
SCHEMBL17268092 0.87 KLKB1 (0.61) KLKB1KLK1PSMB1PSMB9PSMB10
SCHEMBL14485405 0.86 KLKB1 (0.64) KLKB1KLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2729443-B3 BENZYLAMINE DERIVATIVES AS INHIBITORS OF PLASMA KALLIKREIN KALVISTA PHARMACEUTICALS LTD (GB) 2020-02-12 EP disclosed