SCHEMBL21686097

SCHEMBL21686097

COc1cc(-c2nc(-c3c(C)c(Cl)c(C)[n+](O)c3C)no2)cc([N+](=O)[O-])c1O

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
COMT P21964 1/20 0.64
NPC1 O15118 1/20 0.44
HPGD P15428 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
POLB P06746 11/20 0.43
TP53 P04637 4/20 0.43
S1PR1 P21453 2/20 0.42
MAPT P10636 8/20 0.42
CSNK2A2 P19784 1/20 0.39
CSNK2B P67870 1/20 0.39
CSNK2A1 P68400 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21686045 0.94 COMT (0.68) COMTNPC1HPGDRAB9ASMN1; SMN2
SCHEMBL15019301 0.90 COMT (0.79) COMTNPC1HPGDRAB9ASMN1; SMN2
SCHEMBL3591312 0.85 COMT (0.55) COMTNPC1HPGDRAB9ASMN1; SMN2
SCHEMBL30471666 0.85 COMT (0.55) COMTNPC1HPGDRAB9ASMN1; SMN2
SCHEMBL20614242 0.82 COMT (0.85) COMTNPC1HPGDRAB9ASMN1; SMN2
SCHEMBL21388412 0.82 COMT (0.52) COMTNPC1HPGDRAB9ASMN1; SMN2
SCHEMBL30590323 0.81 COMT (0.74) COMTNPC1HPGDRAB9ASMN1; SMN2
SCHEMBL22578262 0.80 COMT (0.70) COMTNPC1HPGDRAB9ASMN1; SMN2
SCHEMBL26135190 0.79 COMT (0.74) COMTNPC1HPGDRAB9ASMN1; SMN2
Ammonia Solution, Strong SCHEMBL30590378 0.79 COMT (0.73) COMTNPC1HPGDRAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3604299-B1 CHEMICAL COMPOUND USEFUL AS INTERMEDIATE FOR PREPARING A CATECHOL-0-METHYL TRANSFERASE INHIBITOR BIAL PORTELA & CA SA (PT) 2023-07-26 EP disclosed
EP-3604299-A1 CHEMICAL COMPOUND USEFUL AS INTERMEDIATE FOR PREPARING A CATECHOL-0-METHYL TRANSFERASE INHIBITOR Bial-Portela & CA, S.A. (PT) 2020-02-05 EP disclosed