SCHEMBL21709197

SCHEMBL21709197

c1ccc(-c2ccc(-n3c4cc(-c5cccc(-c6ccccc6)c5)ccc4c4c5ccccc5ccc43)cc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 2/20 0.37
CYP1B1 Q16678 1/20 0.37
KDM4E B2RXH2 1/20 0.35
ATM Q13315 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
LDHA P00338 1/20 0.35
MAOB P27338 1/20 0.35
MEN1 O00255 1/20 0.35
HSP90AA1 P07900 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35
NR3C1 P04150 1/20 0.35
TDP1 Q9NUW8 1/20 0.34
CYP1A2 P05177 1/20 0.34
FYN P06241 1/20 0.34
MAPK3 P27361 1/20 0.34
AHR P35869 1/20 0.34
PAX8 Q06710 1/20 0.34
ABCG2 Q9UNQ0 1/20 0.34
CDK4 P11802 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13589073 0.97 KDM4E (0.35) CYP1A1CYP1B1KDM4EATML3MBTL1
SCHEMBL21709192 0.97 ATM (0.37) CYP1A1CYP1B1KDM4EATML3MBTL1
SCHEMBL13309509 0.97 ATM (0.37) CYP1A1CYP1B1KDM4EATML3MBTL1
SCHEMBL15739332 0.94 EGFR (0.37) CYP1A1CYP1B1MAOBMEN1HSP90AA1
SCHEMBL22483177 0.93 ESR1 (0.38) CYP1A1CYP1B1KDM4EATML3MBTL1
SCHEMBL22483173 0.93 ESR1 (0.38) CYP1A1CYP1B1KDM4EATML3MBTL1
SCHEMBL17642164 0.93 ATM (0.40) CYP1A1KDM4EATML3MBTL1LDHA
SCHEMBL15739329 0.91 EGFR (0.40) CYP1A1CYP1B1KDM4EATML3MBTL1
SCHEMBL14182858 0.91 MCL1 (0.39) CYP1A1CYP1B1KDM4EATML3MBTL1
SCHEMBL15860077 0.91 AVPR1A (0.35) CYP1A1CYP1B1KDM4EATML3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020032424-A1 ORGANIC ELECTRONIC ELEMENT COMPRISING, AS HOST MATERIAL, MIXTURE OF DIFFERENT KINDS OF COMPOUNDS, AND ELECTRONIC DEVICE THEREOF 덕산네오룩스 주식회사 2020-02-13 WO disclosed
WO-2020032447-A1 ORGANIC ELECTRONIC ELEMENT COMPRISING, AS HOST MATERIAL, MIXTURE OF DIFFERENT KINDS OF COMPOUNDS, AND ELECTRONIC DEVICE THEREOF 덕산네오룩스 주식회사 2020-02-13 WO disclosed