SCHEMBL21733591

SCHEMBL21733591

Cc1cc(N)nc(C2CCc3c(ncnc3N3CCN(C)CC3)C2)c1C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KRAS P01116 8/20 0.37
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
KDM4E B2RXH2 1/20 0.33
CYP1A2 P05177 2/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2D6 P10635 2/20 0.32
CYP2C19 P33261 2/20 0.32
CNR2 P34972 1/20 0.32
USP2 O75604 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
HIF1A Q16665 1/20 0.32
PIK3CA P42336 1/20 0.32
MTOR P42345 1/20 0.32
HRH4 Q9H3N8 2/20 0.32
RPS6KB1 P23443 1/20 0.31
AKT1 P31749 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21722224 0.91 KRAS (0.35) KRASCYP1A2CYP3A4CYP2C19ALDH1A1
SCHEMBL30178155 0.87 KRAS (0.54) KRAS
SCHEMBL30178153 0.87 KRAS (0.54) KRAS
SCHEMBL30177789 0.87 KRAS (0.54) KRAS
SCHEMBL21733863 0.87 KRAS (0.54) KRAS
SCHEMBL21733588 0.87 KRAS (0.54) KRAS
SCHEMBL21733416 0.87 KRAS (0.54) KRAS
SCHEMBL29191281 0.74 KRAS (0.45) KRASKMT2AMEN1CYP1A2CYP3A4
SCHEMBL21734049 0.73 RPS6KB1 (0.34) KRASCYP1A2CYP3A4CYP2C19ALDH1A1
SCHEMBL30834508 0.73 RPS6KB1 (0.34) KRASCYP1A2CYP3A4CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020035031-A1 FUSED RING COMPOUNDS GENENTECH, INC. (US) 2020-02-20 WO disclosed