SCHEMBL21744541

SCHEMBL21744541

NC(=O)NC/C=C/CN(CC1Cc2ncccc2CN1)[C@H]1CCCc2cccnc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 19/20 1.00
CXCR4 P61073 11/20 0.86
CYP3A4 P08684 9/20 0.86
CHRM3 P20309 1/20 0.65
CHRM2 P08172 1/20 0.62
ADRA2A P08913 1/20 0.62
DRD2 P14416 1/20 0.62
ADRA2C P18825 1/20 0.62
CHRNA7 P36544 1/20 0.62
OPRK1 P41145 1/20 0.62
KCNH2 Q12809 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21744184 1.00 CYP2D6 (1.00) CYP2D6CXCR4CYP3A4CHRM3CHRM2
SCHEMBL21744539 0.93 CYP2D6 (1.00) CYP2D6CXCR4CYP3A4CHRM3
SCHEMBL21743999 0.90 CYP2D6 (0.81) CYP2D6CXCR4CYP3A4CHRM3CHRM2
SCHEMBL21743997 0.89 CYP2D6 (0.80) CYP2D6CXCR4CYP3A4CHRM3CHRM2
SCHEMBL21744819 0.87 CYP2D6 (1.00) CYP2D6CXCR4CYP3A4CHRM3CHRM2
SCHEMBL21744508 0.87 CYP2D6 (1.00) CYP2D6CXCR4CYP3A4CHRM3CHRM2
SCHEMBL21744346 0.87 CYP2D6 (1.00) CYP2D6CXCR4CYP3A4CHRM3CHRM2
SCHEMBL21744661 0.87 CYP2D6 (1.00) CYP2D6CXCR4CYP3A4CHRM3CHRM2
SCHEMBL21744347 0.83 CYP2D6 (0.71) CYP2D6CXCR4CYP3A4CHRM3CHRM2
SCHEMBL21744507 0.79 CYP2D6 (1.00) CYP2D6CXCR4CYP3A4CHRM3CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230112832-A1 Chemokine CXCR4 Receptor Modulators and Uses Related Thereto UNIV EMORY (US) 2023-04-13 US disclosed
US-20200054623-A1 Chemokine CXCR4 Receptor Modulators and Uses Related Thereto EMORY UNIVERSITY 2020-02-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200054623-A1 Chemokine CXCR4 Receptor Modulators and Uses Related Thereto CXCR4, CXCL12, CXCR1 CYP2D6 4404/4885CXCR4 1/4885CYP3A4 4527/4885
US-20230112832-A1 Chemokine CXCR4 Receptor Modulators and Uses Related Thereto CXCR4, CXCL12, CXCR1 CYP2D6 4404/4885CXCR4 1/4885CYP3A4 4527/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.