SCHEMBL21757641

SCHEMBL21757641

CC1(NC=O)CCOc2ccc(F)cc21

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 5/20 0.51
AKR1B10 O60218 1/20 0.48
MAPT P10636 1/20 0.48
AKR1A1 P14550 1/20 0.48
RARA P10276 3/20 0.35
RARB P10826 3/20 0.35
RARG P13631 3/20 0.35
FABP6 P51161 1/20 0.35
KMT2A Q03164 1/20 0.35
APP P05067 2/20 0.34
BACE1 P56817 2/20 0.34
KIF11 P52732 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21757599 0.80 KMT2A (0.36) AKR1B1RARARARBRARGKMT2A
SCHEMBL12188672 0.76 AKR1B1 (0.57) AKR1B1AKR1B10MAPTAKR1A1RARA
SCHEMBL3424941 0.75 AKR1B1 (0.51) AKR1B1AKR1B10MAPTAKR1A1RARA
SCHEMBL17729307 0.73 AKR1B1 (0.55) AKR1B1AKR1B10MAPTAKR1A1RARA
SCHEMBL21757625 0.72 HDAC4 (0.33)
SCHEMBL12257631 0.71 AKR1B1 (0.52) AKR1B1AKR1B10MAPTAKR1A1RARA
SCHEMBL12691918 0.71 AKR1B1 (0.52) AKR1B1AKR1B10MAPTAKR1A1RARA
SCHEMBL30353231 0.71 AKR1B1 (0.55) AKR1B1AKR1B10MAPTAKR1A1FABP6
SCHEMBL12691756 0.70 AKR1B1 (0.51) AKR1B1AKR1B10MAPTAKR1A1RARA
SCHEMBL13183293 0.69 AKR1B1 (0.56) AKR1B1AKR1B10MAPTAKR1A1RARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3215509-B1 SUBSTITUTED PYRROLO[1,2-A]PYRIMIDINES AND THEIR USE IN THE TREATMENT OF MEDICAL DISORDERS LYSOSOMAL THERAPEUTICS INC (US) 2020-02-26 EP disclosed