SCHEMBL2176046

SCHEMBL2176046

Nc1cc(N)nc(C2CCCCC2)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.44
CHRM3 P20309 3/20 0.41
PDE4A P27815 3/20 0.41
PDE4B Q07343 3/20 0.41
PDE4C Q08493 3/20 0.41
PDE4D Q08499 3/20 0.41
HRH4 Q9H3N8 3/20 0.40
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
ALDH1A1 P00352 1/20 0.39
TDO2 P48775 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
GFER P55789 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
POLB P06746 1/20 0.37
CASP3 P42574 1/20 0.37
SENP7 Q9BQF6 1/20 0.37
SENP6 Q9GZR1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16789827 0.88 PDE10A (0.42) BACE1CHRM3PDE4APDE4BPDE4C
SCHEMBL21249496 0.86 BACE1 (0.39) BACE1CHRM3PDE4APDE4BPDE4C
SCHEMBL21249492 0.86 BACE1 (0.39) BACE1CHRM3PDE4APDE4BPDE4C
SCHEMBL15103644 0.84 BACE1 (0.37) BACE1CHRM3PDE4APDE4BPDE4C
SCHEMBL21249439 0.82 HRH4 (0.55) CHRM3PDE4APDE4BPDE4CPDE4D
SCHEMBL24821652 0.79 PDE10A (0.38) BACE1CHRM3PDE4APDE4BPDE4C
SCHEMBL15103604 0.79 BACE1 (0.33) BACE1CHRM3PDE4APDE4BPDE4C
SCHEMBL2403564 0.78 HRH4 (0.50) HRH4ALDH1A1MAPT
SCHEMBL6396181 0.77 CHRM3 (0.43) CHRM3PDE4APDE4BPDE4CPDE4D
SCHEMBL2034798 0.77 CHEK1 (0.47) HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079343-A2 SUBSTITUTED PYRIDINES AND PYRIMIDINES TECHNISCHE UNIVERSITAET WIEN (AT) 2011-07-07 WO disclosed