SCHEMBL21770697

SCHEMBL21770697

CSc1ncc2c(n1)N(C)CCN(c1cccc(CCN(C)C(C)=O)c1)C2=O

nearest known ligand 0.57

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 20/20 0.57
SLC6A2 P23975 13/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20970770 0.93 CACNA2D1 (0.60) CACNA2D1SLC6A2
SCHEMBL19553187 0.89 CACNA2D1 (0.54) CACNA2D1SLC6A2
SCHEMBL21747636 0.88 CACNA2D1 (0.61) CACNA2D1SLC6A2
SCHEMBL19553247 0.87 CACNA2D1 (0.61) CACNA2D1SLC6A2
SCHEMBL21747610 0.86 CACNA2D1 (0.59) CACNA2D1SLC6A2
SCHEMBL21747666 0.85 CACNA2D1 (0.55) CACNA2D1SLC6A2
SCHEMBL19553071 0.84 CACNA2D1 (0.56) CACNA2D1SLC6A2
SCHEMBL21770650 0.84 CACNA2D1 (0.62) CACNA2D1SLC6A2
SCHEMBL21770225 0.84 CACNA2D1 (0.64) CACNA2D1SLC6A2
SCHEMBL21747602 0.83 CACNA2D1 (0.57) CACNA2D1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3452475-B1 TETRAHYDROPYRIMIDODIAZEPINE AND TETRAHYDROPYRIDODIAZEPINE COMPOUNDS FOR TREATING PAIN AND PAIN RELATED CONDITIONS ESTEVE PHARMACEUTICALS SA (ES) 2020-02-26 EP disclosed