SCHEMBL21770900

SCHEMBL21770900

CCC(C)c1ncc2c(n1)N(C)CCN(c1cccc(-c3nnc(C)o3)c1)C2=O

nearest known ligand 0.74

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 20/20 0.74
CACNA2D2 Q9NY47 1/20 0.72
SLC6A2 P23975 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19564721 0.85 CACNA2D1 (1.00) CACNA2D1CACNA2D2SLC6A2
SCHEMBL19553337 0.84 CACNA2D1 (1.00) CACNA2D1CACNA2D2SLC6A2
SCHEMBL19552875 0.84 CACNA2D1 (0.83) CACNA2D1CACNA2D2SLC6A2
SCHEMBL19552934 0.83 CACNA2D1 (1.00) CACNA2D1CACNA2D2SLC6A2
SCHEMBL19553540 0.83 CACNA2D1 (0.79) CACNA2D1CACNA2D2SLC6A2
SCHEMBL21770910 0.81 CACNA2D1 (0.53) CACNA2D1SLC6A2
SCHEMBL19553157 0.80 CACNA2D1 (0.83) CACNA2D1CACNA2D2SLC6A2
SCHEMBL19553084 0.80 CACNA2D1 (0.74) CACNA2D1CACNA2D2SLC6A2
SCHEMBL19552884 0.79 CACNA2D1 (0.81) CACNA2D1CACNA2D2
SCHEMBL19553307 0.79 CACNA2D1 (0.70) CACNA2D1CACNA2D2SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3452475-B1 TETRAHYDROPYRIMIDODIAZEPINE AND TETRAHYDROPYRIDODIAZEPINE COMPOUNDS FOR TREATING PAIN AND PAIN RELATED CONDITIONS ESTEVE PHARMACEUTICALS SA (ES) 2020-02-26 EP disclosed