SCHEMBL21779429

SCHEMBL21779429

NC(=O)c1cc(-c2ccc(F)cc2)cnc1N

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CB P42338 1/20 0.58
MAP4K4 O95819 3/20 0.57
CHRNA7 P36544 2/20 0.53
IKBKB O14920 2/20 0.52
CHUK O15111 2/20 0.52
CHEK2 O96017 3/20 0.50
FYN P06241 3/20 0.48
MKNK1 Q9BUB5 1/20 0.48
BMPR1B O00238 1/20 0.47
BMPR1A P36894 1/20 0.47
TGFBR1 P36897 1/20 0.47
ACVRL1 P37023 1/20 0.47
ACVR1 Q04771 1/20 0.47
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45
CSF1R P07333 1/20 0.44
IKBKE Q14164 1/20 0.44
TBK1 Q9UHD2 1/20 0.44
EIF2S1 P05198 1/20 0.44
EIF2AK3 Q9NZJ5 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18617182 0.85 CHEK2 (0.64) PIK3CBMAP4K4CHEK2FYNMKNK1
SCHEMBL18615835 0.85 CHEK2 (0.64) PIK3CBMAP4K4IKBKBCHUKCHEK2
SCHEMBL18615844 0.84 PIK3CB (0.67) PIK3CBMAP4K4CHRNA7CHEK2FYN
SCHEMBL18615848 0.83 MKNK1 (0.61) PIK3CBMAP4K4IKBKBCHUKCHEK2
SCHEMBL18615823 0.83 MAP4K4 (0.60) PIK3CBMAP4K4IKBKBCHEK2FYN
SCHEMBL18616649 0.83 MAP4K4 (0.62) PIK3CBMAP4K4CHEK2FYNMKNK1
SCHEMBL18616283 0.82 PIK3CB (0.68) PIK3CBIKBKBCHUKCHEK2IKBKE
SCHEMBL18616712 0.81 PIK3CB (0.56) PIK3CBMAP4K4CHRNA7IKBKBCHEK2
SCHEMBL18617207 0.80 PIK3CB (0.58) PIK3CBMAP4K4CHRNA7IKBKBCHEK2
SCHEMBL18616321 0.80 PIK3CB (0.58) PIK3CBMAP4K4CHRNA7CHEK2FYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3344613-B1 HETEROARYL COMPOUNDS AND THEIR USE AS THERAPEUTIC DRUGS DONG A SOCIO HOLDINGS CO LTD (KR) 2020-03-04 EP disclosed