SCHEMBL21780941

SCHEMBL21780941

Cc1ccc(OCCN2CCC(CF)C2)cc1

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.56
ESR1 P03372 7/20 0.49
LTA4H P09960 2/20 0.48
KDM1A O60341 2/20 0.47
KDM4E B2RXH2 1/20 0.47
SIGMAR1 Q99720 2/20 0.47
TMEM97 Q5BJF2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21780738 0.88 KDM1A (0.54) HRH3ESR1KDM1A
SCHEMBL17845116 0.86 ESR1 (0.49) ESR1LTA4HKDM4ESIGMAR1TMEM97
SCHEMBL17845086 0.86 ESR1 (0.49) ESR1LTA4HKDM4ESIGMAR1TMEM97
SCHEMBL17845197 0.86 ESR1 (0.59) ESR1LTA4H
SCHEMBL17845198 0.86 ESR1 (0.59) ESR1LTA4H
SCHEMBL21780869 0.86 TMEM97 (0.63) ESR1LTA4HKDM1ASIGMAR1TMEM97
SCHEMBL23474881 0.85 KDM4E (0.60) HRH3ESR1LTA4HKDM4E
SCHEMBL23474993 0.85 MEN1 (0.52) ESR1LTA4HKDM4ESIGMAR1TMEM97
SCHEMBL23474962 0.85 KDM4E (0.60) HRH3ESR1LTA4HKDM4E
SCHEMBL23474994 0.85 KDM4E (0.60) HRH3ESR1LTA4HKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233828-B1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF HOFFMANN LA ROCHE (CH) 2020-03-04 EP disclosed