SCHEMBL21782121

SCHEMBL21782121

CCC(C)C(C(CC(=O)N1CCCC1C(OC)C(C)C(=O)NC(Cc1ccccc1)C(=O)NCc1ccc(NC(=O)C(CCCNC)NC(=O)CNC(=O)CCC(=O)N2CCCCC2)cc1)OC)N(C)C(=O)CNC

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.43
FOLH1 Q04609 3/20 0.39
AKT1 P31749 3/20 0.37
TTR P02766 2/20 0.35
PSMB8 P28062 1/20 0.35
PSMB5 P28074 1/20 0.35
ITGB1 P05556 1/20 0.33
ITGA5 P08648 1/20 0.33
SSTR2 P30874 1/20 0.33
REN P00797 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
LCK P06239 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21781779 0.87 CYP3A4 (0.42) CYP3A4FOLH1AKT1TTRITGB1
SCHEMBL21782123 0.87 CYP3A4 (0.45) CYP3A4FOLH1AKT1TTRITGB1
SCHEMBL21781954 0.86 CYP3A4 (0.44) CYP3A4FOLH1AKT1TTRSSTR2
SCHEMBL21781773 0.83 CYP3A4 (0.45) CYP3A4FOLH1AKT1TTRSSTR2
SCHEMBL21781950 0.83 CYP3A4 (0.46) CYP3A4FOLH1AKT1TTRSSTR2
SCHEMBL24136561 0.82 CYP3A4 (0.46) CYP3A4FOLH1AKT1TTRSSTR2
SCHEMBL21781872 0.82 CYP3A4 (0.46) CYP3A4FOLH1AKT1TTRSSTR2
SCHEMBL21781961 0.82 CYP3A4 (0.46) CYP3A4FOLH1AKT1TTRSSTR2
SCHEMBL21781997 0.82 CYP3A4 (0.45) CYP3A4FOLH1AKT1TTRSSTR2
SCHEMBL24136571 0.80 CYP3A4 (0.46) CYP3A4FOLH1AKT1TTRSSTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3617221-A1 CYTOTOXIN AND CONJUGATE, USES OF SAME, AND PREPARATION METHOD THEREFOR Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd. (CN) 2020-03-04 EP disclosed