SCHEMBL21783175

SCHEMBL21783175

Cc1c(N2C[C@@H](C)N[C@@H](C)C2)c(F)c2c(c1NC(=O)OC(C)(P(=O)(O)O)P(=O)(O)O)c(=O)c(C(=O)O)cn2C1CC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.61
KMT2A Q03164 1/20 0.61
KCNH2 Q12809 4/20 0.57
POLB P06746 2/20 0.57
CACNA1F O60840 1/20 0.57
MAPK1 P28482 1/20 0.57
CACNA1D Q01668 1/20 0.57
CACNA1S Q13698 1/20 0.57
CACNA1C Q13936 1/20 0.57
HRH3 Q9Y5N1 1/20 0.43
GSK3B P49841 10/20 0.41
TOP2A P11388 2/20 0.41
TOP2B Q02880 2/20 0.41
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
HPGD P15428 2/20 0.40
PRKD3 O94806 1/20 0.40
ALOX15 P16050 1/20 0.40
OPRM1 P35372 1/20 0.40
CLK2 P49760 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21074643 0.94 MEN1 (0.65) MEN1KMT2AKCNH2POLBCACNA1F
SCHEMBL21074712 0.81 MEN1 (0.67) MEN1KMT2AKCNH2POLBCACNA1F
SCHEMBL21074751 0.81 KDM4E (0.58) MEN1KMT2AKCNH2POLBCACNA1F
SCHEMBL21074635 0.79 POLB (0.54) MEN1KMT2AKCNH2POLBCACNA1F
SCHEMBL21074775 0.78 MEN1 (0.65) MEN1KMT2AKCNH2POLBCACNA1F
SCHEMBL10584006 0.78 MEN1 (0.86) MEN1KMT2AKCNH2POLBCACNA1F
SCHEMBL10584011 0.78 MEN1 (0.86) MEN1KMT2AKCNH2POLBCACNA1F
Orbifloxacin SCHEMBL29420860 0.77 MEN1 (1.00) MEN1KMT2AKCNH2POLBCACNA1F
Orbifloxacin SCHEMBL9374152 0.77 MEN1 (1.00) MEN1KMT2AKCNH2POLBCACNA1F
Orbifloxacin SCHEMBL125116 0.77 MEN1 (1.00) MEN1KMT2AKCNH2POLBCACNA1F

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020014269-A9 BISPHOSPHONATE QUINOLONE CONJUGATES AND USES THEREOF BIOVINC, LLC. (US) 2020-03-05 WO disclosed