SCHEMBL21783299

SCHEMBL21783299

COc1c(N2C[C@@H](C)C[C@H](N)C2)ccc2c(=O)c(C(=O)OC(Cc3cccnc3)(P(=O)(O)O)P(=O)(O)O)cn(C3CC3)c12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.44
CYP3A4 P08684 1/20 0.36
PIM2 Q9P1W9 6/20 0.34
GSK3B P49841 1/20 0.34
KDM4E B2RXH2 3/20 0.34
ALDH1A1 P00352 2/20 0.34
POLB P06746 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
LMNA P02545 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
PIM1 P11309 1/20 0.33
PIM3 Q86V86 1/20 0.33
TOP2A P11388 1/20 0.32
TOP2B Q02880 1/20 0.32
PRKD3 O94806 1/20 0.32
HPGD P15428 1/20 0.32
ALOX15 P16050 1/20 0.32
OPRM1 P35372 1/20 0.32
CLK2 P49760 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21783241 0.86 KCNH2 (0.50) KCNH2CYP3A4GSK3BKDM4EALDH1A1
SCHEMBL21783240 0.85 KCNH2 (0.42) KCNH2CYP3A4PIM2GSK3BKDM4E
SCHEMBL21783296 0.84 KCNH2 (0.50) KCNH2CYP3A4GSK3BKDM4EALDH1A1
SCHEMBL13866591 0.80 KCNH2 (0.56) KCNH2CYP3A4GSK3BKDM4EALDH1A1
Nemonoxacin SCHEMBL2106812 0.78 KCNH2 (0.66) KCNH2CYP3A4GSK3BKDM4EALDH1A1
Nemonoxacin SCHEMBL1006373 0.78 KCNH2 (0.66) KCNH2CYP3A4GSK3BKDM4EALDH1A1
Nemonoxacin SCHEMBL31574403 0.78 KCNH2 (0.66) KCNH2CYP3A4GSK3BKDM4EALDH1A1
SCHEMBL2601623 0.78 KCNH2 (0.59) KCNH2CYP3A4GSK3BKDM4EALDH1A1
Nemonoxacin SCHEMBL14381001 0.78 KCNH2 (0.66) KCNH2CYP3A4GSK3BKDM4EALDH1A1
Nemonoxacin SCHEMBL31574404 0.78 KCNH2 (0.66) KCNH2CYP3A4GSK3BKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020014269-A9 BISPHOSPHONATE QUINOLONE CONJUGATES AND USES THEREOF BIOVINC, LLC. (US) 2020-03-05 WO disclosed