SCHEMBL21783504

SCHEMBL21783504

Cc1nc(S(=O)(=O)Nc2ccon2)c(F)cc1N

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SCN1A P35498 3/20 0.53
SCN8A Q9UQD0 3/20 0.53
SCN5A Q14524 2/20 0.52
SCN9A Q15858 17/20 0.40
CYP2C9 P11712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL21955515 0.99 SCN1A (0.52) SCN1ASCN8ASCN5ASCN9ACYP2C9
SCHEMBL28556000 0.82 SCN1A (0.49) SCN1ASCN8ASCN5ASCN9ACYP2C9
SCHEMBL21777479 0.81 SCN8A (0.57) SCN1ASCN8ASCN5ASCN9A
SCHEMBL31017728 0.79 SCN1A (0.47) SCN1ASCN8ASCN5ASCN9ACYP2C9
SCHEMBL21783416 0.75 SCN1A (0.55) SCN1ASCN8ASCN5ASCN9A
SCHEMBL21783429 0.75 SCN1A (0.58) SCN1ASCN8ASCN5ASCN9ACYP2C9
Hydrochloric Acid SCHEMBL30045377 0.74 SCN1A (0.57) SCN1ASCN8ASCN5ASCN9ACYP2C9
Hydrochloric Acid SCHEMBL21955494 0.74 SCN1A (0.57) SCN1ASCN8ASCN5ASCN9ACYP2C9
Hydrochloric Acid SCHEMBL21955493 0.73 SCN1A (0.56) SCN1ASCN8ASCN5ASCN9ACYP2C9
SCHEMBL21783509 0.72 BACE1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11639351-B2 Heteroaryl-substituted sulfonamide compounds and their use as therapeutic agents XENON PHARMACEUTICALS INC. 2023-05-02 US disclosed
US-10981905-B2 Heteroaryl-substituted sulfonamide compounds and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2021-04-20 US disclosed
US-20200157089-A1 HETEROARYL-SUBSTITUTED SULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2020-05-21 US disclosed
WO-2020047323-A1 HETEROARYL-SUBSTITUTED SULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2020-03-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11639351-B2 Heteroaryl-substituted sulfonamide compounds and their use as therapeutic agents SCN1A, SCN2A, SCN2B SCN1A 1/4885SCN8A 6/4885SCN5A 7/4885
US-20200157089-A1 HETEROARYL-SUBSTITUTED SULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS SCN1A, SCN2A, SCN2B SCN1A 1/4885SCN8A 6/4885SCN5A 7/4885
US-10981905-B2 Heteroaryl-substituted sulfonamide compounds and their use as therapeutic agents SCN1A, SCN2A, SCN2B SCN1A 1/4885SCN8A 6/4885SCN5A 7/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.