SCHEMBL21784359

SCHEMBL21784359

O=C(I)NCCCCN(Cc1nc2ccccc2[nH]1)[C@H]1CCCc2cccnc21

nearest known ligand 0.78

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 20/20 0.78
CHRM2 P08172 1/20 0.73
CYP2D6 P10635 1/20 0.73
DRD2 P14416 1/20 0.73
OPRM1 P35372 1/20 0.73
KCNH2 Q12809 1/20 0.73
CYP3A4 P08684 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2513431 0.92 CXCR4 (0.78) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL2508668 0.92 CXCR4 (0.80) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL2513427 0.92 CXCR4 (0.78) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL2508662 0.92 CXCR4 (0.80) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL2526582 0.91 CXCR4 (0.75) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL14131181 0.91 CXCR4 (0.75) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL2508580 0.90 CXCR4 (0.77) CXCR4CHRM2CYP2D6DRD2OPRM1
Bromide SCHEMBL5134127 0.90 CXCR4 (0.74) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL14131218 0.89 CXCR4 (0.73) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL2510374 0.89 CXCR4 (0.78) CXCR4CHRM2CYP2D6DRD2OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020047410-A1 COMPOSITIONS OF CXCR4 INHIBITORS AND METHODS OF PREPARATION AND USE X4 PHARMACEUTICALS, INC. (US) 2020-03-05 WO disclosed