SCHEMBL2180707

SCHEMBL2180707

NS(=O)(=O)c1cccc(CNc2nccn3c(-c4ccc(O)cc4)cnc23)c1

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TTK P33981 12/20 0.52
PI4KB Q9UBF8 1/20 0.51
NTRK1 P04629 1/20 0.44
NTRK3 Q16288 1/20 0.44
NTRK2 Q16620 1/20 0.44
ADORA3 P0DMS8 5/20 0.41
FLT3 P36888 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12409445 0.91 PI4KB (0.60) TTKPI4KBADORA3
SCHEMBL12409266 0.89 PI4KB (0.63) TTKPI4KBNTRK1NTRK3NTRK2
SCHEMBL2181894 0.88 TTK (0.53) TTK
SCHEMBL2178599 0.88 TTK (0.48) TTKPI4KBNTRK1NTRK3NTRK2
SCHEMBL12409263 0.87 PI4KB (0.51) TTKPI4KBADORA3
SCHEMBL14668730 0.86 TTK (0.56) TTKADORA3
SCHEMBL14664246 0.85 PI4KB (0.53) TTKPI4KBNTRK1NTRK3NTRK2
SCHEMBL12409495 0.84 PI4KB (0.44) TTKPI4KBNTRK1NTRK3NTRK2
SCHEMBL12409438 0.83 TTK (0.44) TTKADORA3FLT3
SCHEMBL12409437 0.83 TTK (0.47) TTKPI4KBADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2567960-A2 Imidazo[1,2-a]pyrazine compounds for treatment of viral infections such as hepatitis Biofocus DPI Limited (GB) 2013-03-13 EP disclosed
EP-2193131-B1 IMIDAZO[1,2-A]PYRAZINE COMPOUNDS FOR TREATMENT OF VIRAL INFECTIONS SUCH AS HEPATITIS BIOFOCUS DPI LTD (GB) 2013-01-30 EP disclosed
US-8362018-B2 Substituted imidazo[1,2-a]pyrazine compounds useful for the treatment of viral infections BIOFOCUS DPI, LTD. (GB) 2013-01-29 US disclosed
US-8362018-B2 Substituted imidazo[1,2-a]pyrazine compounds useful for the treatment of viral infections BIOFOCUS DPI, LTD. (GB) 2013-01-29 US disclosed
US-8362018-B2 Substituted imidazo[1,2-a]pyrazine compounds useful for the treatment of viral infections BIOFOCUS DPI, LTD. (GB) 2013-01-29 US disclosed
US-20110166147-A1 IMIDAZOPYRAZINE COMPOUNDS BIOFOCUS DPI, LTD. (GB) 2011-07-07 US disclosed
US-20110166147-A1 IMIDAZOPYRAZINE COMPOUNDS BIOFOCUS DPI, LTD. (GB) 2011-07-07 US disclosed
EP-2193131-A2 IMIDAZO[1,2-A]PYRAZINE COMPOUNDS FOR TREATMENT OF VIRAL INFECTIONS SUCH AS HEPATITIS Biofocus DPI Limited (GB) 2010-06-09 EP disclosed
WO-2009024585-A2 IMIDAZO [1,2-A] PYRAZINE COMPOUNDS FOR TREATMENT OF VIRAL INFECTIONS SUCH AS HEPATITIS BIOFOCUS DPI LIMITED (GB) 2009-02-26 WO disclosed
WO-2009024585-A2 IMIDAZO [1,2-A] PYRAZINE COMPOUNDS FOR TREATMENT OF VIRAL INFECTIONS SUCH AS HEPATITIS BIOFOCUS DPI LIMITED (GB) 2009-02-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110166147-A1 IMIDAZOPYRAZINE COMPOUNDS CYP3A5, HAVCR2, CYP3A43 TTK 3239/4885PI4KB 2534/4885NTRK1 3339/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.