SCHEMBL21809409

SCHEMBL21809409

O=C(NCCc1c[nH]c2ccc(F)cc12)c1cc(Cc2ccc(F)cc2F)on1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.56
MTNR1A P48039 1/20 0.56
MTNR1B P49286 1/20 0.56
SNCA P37840 8/20 0.54
TRPV1 Q8NER1 1/20 0.54
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
SPR P35270 1/20 0.52
MPO P05164 5/20 0.50
SLC6A4 P31645 2/20 0.50
SIRT1 Q96EB6 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30487840 1.00 NOTUM (0.56) NOTUMMTNR1AMTNR1BSNCATRPV1
SCHEMBL30487839 1.00 NOTUM (0.56) NOTUMMTNR1AMTNR1BSNCATRPV1
SCHEMBL30487829 0.93 SNCA (0.56) NOTUMMTNR1AMTNR1BSNCATRPV1
SCHEMBL21809406 0.93 SNCA (0.56) NOTUMMTNR1AMTNR1BSNCATRPV1
SCHEMBL21809405 0.92 SNCA (0.60) NOTUMMTNR1AMTNR1BSNCATRPV1
SCHEMBL30487835 0.92 SNCA (0.60) NOTUMMTNR1AMTNR1BSNCATRPV1
SCHEMBL30487847 0.92 SNCA (0.60) NOTUMMTNR1AMTNR1BSNCATRPV1
SCHEMBL21809408 0.89 SNCA (0.62) NOTUMMTNR1AMTNR1BSNCATRPV1
SCHEMBL21809410 0.89 SNCA (0.57) NOTUMMTNR1AMTNR1BSNCATRPV1
SCHEMBL30487842 0.89 SNCA (0.57) NOTUMMTNR1AMTNR1BSNCATRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12178805-B2 Inhibitors of PDE6Delta for use in the prevention and/or treatment of epilepsy and/or neurodegenerative disorders REMYND N.V. (BE) 2024-12-31 US claimed
US-11939324-B2 Compounds for the treatment of epilepsy, neurodegenerative disorders and other CNS disorders REMYND N.V. (BE) 2024-03-26 US claimed
EP-3621963-B1 COMPOUNDS FOR THE TREATMENT OF EPILEPSY, NEURODEGENERATIVE DISORDERS AND OTHER CNS DISORDERS REMYND N V (BE) 2024-01-24 EP claimed
US-20230099111-A1 COMPOUNDS FOR THE TREATMENT OF EPILEPSY, NEURODEGENERATIVE DISORDERS AND OTHER CNS DISORDERS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2023-03-30 US claimed
US-11548881-B2 Compounds for the treatment of epilepsy, neurodegenerative disorders and other CNS disorders REMYND N.V. (BE) 2023-01-10 US claimed
US-20200253934-A1 INHIBITORS OF PDE6DELTA FOR USE IN THE PREVENTION AND/OR TREATMENT OF EPILEPSY AND/OR NEURODEGENERATIVE DISORDERS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2020-08-13 US claimed
US-20200095238-A1 COMPOUNDS FOR THE TREATMENT OF EPILEPSY, NEURODEGENERATIVE DISORDERS AND OTHER CNS DISORDERS CISTIM (BE) 2020-03-26 US claimed
US-12178805-B2 Inhibitors of PDE6Delta for use in the prevention and/or treatment of epilepsy and/or neurodegenerative disorders REMYND N.V. (BE) 2024-12-31 US disclosed
US-11939324-B2 Compounds for the treatment of epilepsy, neurodegenerative disorders and other CNS disorders REMYND N.V. (BE) 2024-03-26 US disclosed
EP-3621963-B1 COMPOUNDS FOR THE TREATMENT OF EPILEPSY, NEURODEGENERATIVE DISORDERS AND OTHER CNS DISORDERS REMYND N V (BE) 2024-01-24 EP disclosed
EP-3621963-B1 COMPOUNDS FOR THE TREATMENT OF EPILEPSY, NEURODEGENERATIVE DISORDERS AND OTHER CNS DISORDERS REMYND N V (BE) 2024-01-24 EP disclosed
CN-110650955-B Compounds for the treatment of epilepsy, neurodegenerative disorders and other CNS disorders 瑞敏德股份有限公司 2023-07-25 CN disclosed
US-20230099111-A1 COMPOUNDS FOR THE TREATMENT OF EPILEPSY, NEURODEGENERATIVE DISORDERS AND OTHER CNS DISORDERS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2023-03-30 US disclosed
US-11548881-B2 Compounds for the treatment of epilepsy, neurodegenerative disorders and other CNS disorders REMYND N.V. (BE) 2023-01-10 US disclosed
US-11548881-B2 Compounds for the treatment of epilepsy, neurodegenerative disorders and other CNS disorders REMYND N.V. (BE) 2023-01-10 US disclosed
US-20200253934-A1 INHIBITORS OF PDE6DELTA FOR USE IN THE PREVENTION AND/OR TREATMENT OF EPILEPSY AND/OR NEURODEGENERATIVE DISORDERS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2020-08-13 US disclosed
US-20200253934-A1 INHIBITORS OF PDE6DELTA FOR USE IN THE PREVENTION AND/OR TREATMENT OF EPILEPSY AND/OR NEURODEGENERATIVE DISORDERS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2020-08-13 US disclosed
US-20200095238-A1 COMPOUNDS FOR THE TREATMENT OF EPILEPSY, NEURODEGENERATIVE DISORDERS AND OTHER CNS DISORDERS CISTIM (BE) 2020-03-26 US disclosed
CN-110650955-A Compounds for the treatment of epilepsy, neurodegenerative disorders and other CNS disorders 瑞敏德股份有限公司 2020-01-03 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200095238-A1 COMPOUNDS FOR THE TREATMENT OF EPILEPSY, NEURODEGENERATIVE DISORDERS AND OTHER CNS DISORDERS MAPT, PSEN1, PSEN2 NOTUM 1671/4885MTNR1A 86/4885MTNR1B 139/4885
US-12178805-B2 Inhibitors of PDE6Delta for use in the prevention and/or treatment of epilepsy and/or neurodegenerative disorders PDE4A, PDE12, PDE2A NOTUM 2205/4885MTNR1A 1212/4885MTNR1B 1101/4885
US-20230099111-A1 COMPOUNDS FOR THE TREATMENT OF EPILEPSY, NEURODEGENERATIVE DISORDERS AND OTHER CNS DISORDERS MAPT, PSEN1, PSEN2 NOTUM 1671/4885MTNR1A 86/4885MTNR1B 139/4885
US-11548881-B2 Compounds for the treatment of epilepsy, neurodegenerative disorders and other CNS disorders MAPT, PSEN1, PSEN2 NOTUM 1671/4885MTNR1A 86/4885MTNR1B 139/4885
US-20200253934-A1 INHIBITORS OF PDE6DELTA FOR USE IN THE PREVENTION AND/OR TREATMENT OF EPILEPSY AND/OR NEURODEGENERATIVE DISORDERS PDE4A, PDE12, PDE2A NOTUM 2205/4885MTNR1A 1212/4885MTNR1B 1101/4885
US-11939324-B2 Compounds for the treatment of epilepsy, neurodegenerative disorders and other CNS disorders MAPT, PSEN1, PSEN2 NOTUM 1671/4885MTNR1A 86/4885MTNR1B 139/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.