SCHEMBL21843663

SCHEMBL21843663

Cc1ccc2[nH]nc(C#Cc3cncc(C(=O)Nc4ccc(CN5CCN(C)CC5)c(C(F)(F)F)c4)c3)c2c1

nearest known ligand 0.68

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RET P07949 3/20 0.68
FGFR1 P11362 9/20 0.66
KDR P35968 8/20 0.66
KIF5B P33176 1/20 0.63
CCDC6 Q16204 1/20 0.63
ABL1 P00519 8/20 0.59
KIT P10721 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21843573 0.94 RET (0.69) RETFGFR1KDRKIF5BCCDC6
SCHEMBL21843583 0.93 RET (0.68) RETFGFR1KDRKIF5BCCDC6
SCHEMBL21843513 0.93 RET (0.68) RETFGFR1KDRKIF5BCCDC6
SCHEMBL24283331 0.92 RET (0.68) RETFGFR1KDRKIF5BCCDC6
SCHEMBL24283201 0.92 RET (0.67) RETFGFR1KDRKIF5BCCDC6
SCHEMBL21843582 0.91 FGFR1 (0.74) RETFGFR1KDRKIF5BCCDC6
SCHEMBL24283346 0.91 RET (0.66) RETFGFR1KDRKIF5BCCDC6
SCHEMBL21843664 0.91 RET (0.66) RETFGFR1KDRKIF5BCCDC6
SCHEMBL24283334 0.91 RET (0.69) RETFGFR1KDRKIF5BCCDC6
SCHEMBL24283234 0.90 RET (0.65) RETFGFR1KDRKIF5BCCDC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020053812-A1 ALKYNYL NICOTINAMIDE COMPOUNDS AS KINASE INHIBITORS PURDUE RESEARCH FOUNDATION (US) 2020-03-19 WO disclosed