SCHEMBL21851607

SCHEMBL21851607

O=C1c2cc(N3CCN4CCC3CC4)ccc2-c2cccc([N+](=O)[O-])c21

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.47
CHRNA1 P02708 3/20 0.46
CHRNB2 P17787 3/20 0.46
CHRNB4 P30926 3/20 0.46
CHRNA3 P32297 3/20 0.46
CHRNA4 P43681 3/20 0.46
CHRNA7 P36544 3/20 0.46
HTR3A P46098 2/20 0.46
S100A4 P26447 2/20 0.41
PTPRC P08575 1/20 0.39
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
RECQL P46063 1/20 0.38
MCL1 Q07820 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
AURKA O14965 1/20 0.37
ALDH1A1 P00352 1/20 0.36
TP53 P04637 1/20 0.36
CYP1A2 P05177 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21851632 0.83 CHRNA1 (0.58) KCNH2CHRNA1CHRNB2CHRNB4CHRNA3
SCHEMBL21999211 0.82 KCNH2 (0.51) KCNH2CHRNA1CHRNB2CHRNB4CHRNA3
SCHEMBL22522388 0.82 KCNH2 (0.51) KCNH2CHRNA1CHRNB2CHRNB4CHRNA3
SCHEMBL1793080 0.80 KCNH2 (0.62) KCNH2CHRNA1CHRNB2CHRNB4CHRNA3
SCHEMBL21851605 0.79 CHRNA1 (0.49) KCNH2CHRNA1CHRNB2CHRNB4CHRNA3
SCHEMBL17985441 0.77 CHRNA1 (0.72) KCNH2CHRNA1CHRNB2CHRNB4CHRNA3
SCHEMBL21851634 0.73 CHRNA1 (0.65) KCNH2CHRNA1CHRNB2CHRNB4CHRNA3
SCHEMBL21851709 0.73 KCNH2 (0.50) KCNH2CHRNA1CHRNB2CHRNB4CHRNA3
SCHEMBL22522653 0.73 KCNH2 (0.50) KCNH2CHRNA1CHRNB2CHRNB4CHRNA3
SCHEMBL22522390 0.73 KCNH2 (0.50) KCNH2CHRNA1CHRNB2CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3632918-A1 LIGAND COMPOUND OF 7 NICOTINIC ACETYLCHOLINE RECEPTOR AND APPLICATION THEREOF Beijing Normal University (CN) 2020-04-08 EP disclosed