SCHEMBL2185302

SCHEMBL2185302

CCS(=O)(=O)C(NC(=O)c1cncc2c1cnn2-c1ccc(F)cc1)c1ccncc1

nearest known ligand 0.65

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 20/20 0.65
CYP3A4 P08684 1/20 0.65
KCNH2 Q12809 2/20 0.54
ADRB1 P08588 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL568174 0.86 CCR1 (0.76) CCR1CYP3A4KCNH2ADRB1
SCHEMBL566936 0.80 CCR1 (0.61) CCR1CYP3A4KCNH2ADRB1
SCHEMBL567954 0.79 CCR1 (1.00) CCR1CYP3A4KCNH2ADRB1
SCHEMBL568285 0.79 CCR1 (1.00) CCR1CYP3A4KCNH2ADRB1
SCHEMBL567978 0.79 CCR1 (0.84) CCR1CYP3A4KCNH2ADRB1
SCHEMBL568184 0.78 CCR1 (0.89) CCR1CYP3A4KCNH2ADRB1
SCHEMBL567742 0.78 CCR1 (0.70) CCR1CYP3A4KCNH2ADRB1
SCHEMBL567856 0.78 CCR1 (0.88) CCR1CYP3A4KCNH2ADRB1
SCHEMBL568069 0.78 CCR1 (0.80) CCR1CYP3A4KCNH2ADRB1
SCHEMBL567342 0.78 CCR1 (0.67) CCR1CYP3A4KCNH2ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346868-A1 AZAINDAZOLE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-07-27 EP disclosed