SCHEMBL21856767

SCHEMBL21856767

CCn1cc(C#N)c2cc(Oc3ccc(N(C)C(=O)[C@@H]4CCC(=O)N4)cc3)ccc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PFKFB3 Q16875 18/20 1.00
PFKFB1 P16118 16/20 0.76
PFKFB2 O60825 14/20 0.76
ALDH1A1 P00352 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21856933 0.86 PFKFB3 (1.00) PFKFB3PFKFB1PFKFB2
SCHEMBL21856723 0.86 PFKFB3 (1.00) PFKFB3PFKFB1PFKFB2
SCHEMBL28652895 0.84 PFKFB3 (0.78) PFKFB3PFKFB1PFKFB2
SCHEMBL30268345 0.84 PFKFB3 (0.78) PFKFB3PFKFB1PFKFB2
SCHEMBL21856728 0.73 PFKFB3 (1.00) PFKFB3PFKFB1PFKFB2
SCHEMBL21856810 0.72 PFKFB3 (1.00) PFKFB3PFKFB1PFKFB2
SCHEMBL21856796 0.72 PFKFB3 (1.00) PFKFB3PFKFB1PFKFB2
SCHEMBL21856838 0.71 PFKFB3 (1.00) PFKFB3PFKFB1PFKFB2
SCHEMBL21857036 0.70 PFKFB3 (1.00) PFKFB3PFKFB1PFKFB2ALDH1A1
SCHEMBL21856792 0.68 PFKFB3 (1.00) PFKFB3PFKFB1PFKFB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020080979-A1 PFKFB3 INHIBITORS AND THEIR USES GERO DISCOVERY LIMITED LIABILITY COMPANY (RU) 2020-04-23 WO claimed
CN-113396145-A PFKFB3 inhibitors and uses thereof 盖罗发现有限责任公司 2021-09-14 CN disclosed
WO-2020080979-A1 PFKFB3 INHIBITORS AND THEIR USES GERO DISCOVERY LIMITED LIABILITY COMPANY (RU) 2020-04-23 WO disclosed