SCHEMBL2186757

SCHEMBL2186757

CCOC(=O)Oc1c[nH]c2ccccc12

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC22A6 Q4U2R8 2/20 0.65
PKM P14618 1/20 0.57
SMN1; SMN2 Q16637 3/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
MAPT P10636 4/20 0.50
KDM4E B2RXH2 3/20 0.50
ALDH1A1 P00352 3/20 0.50
PBRM1 Q86U86 1/20 0.49
KMT2A Q03164 3/20 0.48
MEN1 O00255 2/20 0.48
ATM Q13315 1/20 0.48
LMNA P02545 2/20 0.47
NR4A2 P43354 1/20 0.45
CREBBP Q92793 1/20 0.45
GABRA1 P14867 1/20 0.45
GABRB2 P47870 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27729377 0.85 SLC22A6 (0.74) SLC22A6SMN1; SMN2MAPTKDM4EALDH1A1
SCHEMBL4624292 0.83 SLC22A6 (0.71) SLC22A6PKMSMN1; SMN2CYP1A2CYP2C19
SCHEMBL352798 0.81 SLC22A6 (0.69) SLC22A6PKMSMN1; SMN2CYP1A2CYP3A4
SCHEMBL148210 0.80 SLC22A6 (0.67) SLC22A6PKMSMN1; SMN2CYP1A2CYP3A4
SCHEMBL28113890 0.80 SLC22A6 (0.67) SLC22A6PKMSMN1; SMN2CYP1A2CYP3A4
SCHEMBL29199780 0.79 SLC22A6 (0.61) SLC22A6PKMSMN1; SMN2CYP1A2CYP3A4
SCHEMBL28747978 0.79 SLC22A6 (0.61) SLC22A6PKMSMN1; SMN2CYP1A2CYP3A4
SCHEMBL29199798 0.79 SLC22A6 (0.61) SLC22A6PKMSMN1; SMN2CYP1A2CYP3A4
Indole Acetate SCHEMBL15553 0.79 SLC22A6 (1.00) SLC22A6PKMSMN1; SMN2CYP1A2CYP2C19
SCHEMBL11350789 0.79 SLC22A6 (0.53) SLC22A6PKMSMN1; SMN2CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2343291-A1 3-(Indolyl)- or 3-(Azaindolyl)-4-arylmaleimide compounds and their use in tumor treatment Johannes Gutenberg-Universität Mainz (DE) 2011-07-13 EP disclosed
EP-0716077-A1 Aromatically substituted omega amino alcanoic acid amides and alcanoic diamides and their use as renine inhibitors CIBA-GEIGY AG (CH) 1996-06-12 EP disclosed
EP-0702004-A2 2,9-diamino- and 2-amino-8-carbamoyl-4-hydroxy-alkanoic acid amid derivatives CIBA-GEIGY AG (CH) 1996-03-20 EP disclosed