SCHEMBL2186906

SCHEMBL2186906

Cc1nnc(C)n1-c1ccc(O[C@@H]2c3cc(Cl)cc(Cl)c3C[C@@H]2N2CCSCC2)c(F)c1

nearest known ligand 0.75

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SLC9A3 P48764 19/20 0.75
CYP2C9 P11712 2/20 0.75
SLC9A5 Q14940 2/20 0.75
CYP2D6 P10635 4/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2189770 1.00 SLC9A3 (0.75) SLC9A3CYP2C9SLC9A5CYP2D6
SCHEMBL2188847 0.92 SLC9A3 (0.78) SLC9A3CYP2C9SLC9A5CYP2D6
SCHEMBL2188843 0.92 SLC9A3 (0.78) SLC9A3CYP2C9SLC9A5CYP2D6
SCHEMBL2186482 0.92 SLC9A3 (0.78) SLC9A3CYP2C9SLC9A5CYP2D6
SCHEMBL2189080 0.90 SLC9A3 (0.75) SLC9A3CYP2C9SLC9A5CYP2D6
SCHEMBL2189085 0.90 SLC9A3 (0.75) SLC9A3CYP2C9SLC9A5CYP2D6
SCHEMBL2261139 0.88 SLC9A3 (0.72) SLC9A3CYP2C9SLC9A5CYP2D6
SCHEMBL2264919 0.88 SLC9A3 (0.77) SLC9A3CYP2C9SLC9A5CYP2D6
SCHEMBL2188477 0.88 SLC9A3 (0.77) SLC9A3CYP2C9SLC9A5CYP2D6
SCHEMBL2261133 0.88 SLC9A3 (0.72) SLC9A3CYP2C9SLC9A5CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2342178-A1 SUBSTITUTED AMINOINDANES AND ANALOGS THEREOF, AND THE PHARMACEUTICAL USE THEREOF Sanofi-Aventis (FR) 2011-07-13 EP claimed
WO-2010025856-A1 SUBSTITUTED AMINOINDANES AND ANALOGS THEREOF, AND THE PHARMACEUTICAL USE THEREOF SANOFI-AVENTIS (FR) 2010-03-11 WO claimed