SCHEMBL21879656

SCHEMBL21879656

Clc1ncc2scc(-c3ccc(OCCBr)cc3)c2n1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTK2 Q05397 5/20 0.39
SYK P43405 1/20 0.34
ATP4A P20648 4/20 0.33
ATP4B P51164 4/20 0.33
RAB9A P51151 3/20 0.33
NPC1 O15118 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MGAM O43451 3/20 0.32
GAA P10253 3/20 0.32
SI P14410 3/20 0.32
MGAM2 Q2M2H8 3/20 0.32
MAPT P10636 2/20 0.32
NPSR1 Q6W5P4 1/20 0.32
HTT P42858 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21953819 0.78 CYSLTR2 (0.42) PTK2SYKRAB9ANPC1HSD17B10
SCHEMBL1674327 0.77 PTK2 (0.44) PTK2SYKRAB9ANPC1SMN1; SMN2
SCHEMBL1682805 0.71 PTK2 (0.45) PTK2SYKRAB9ANPC1SMN1; SMN2
SCHEMBL1682796 0.68 PTK2 (0.50) PTK2SYKRAB9ANPC1SMN1; SMN2
SCHEMBL367112 0.68 SYK (0.41) SYK
SCHEMBL29963047 0.68 SYK (0.41) SYK
SCHEMBL1682843 0.67 PTK2 (0.50) PTK2
SCHEMBL1674220 0.66 SYK (0.39) SYK
SCHEMBL21953511 0.66 SYK (0.38) PTK2SYKSMN1; SMN2MAPTHTT
SCHEMBL29237867 0.65 CYP3A4 (0.47) RAB9ANPC1SMN1; SMN2MGAMGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020085742-A1 HETEROAROMATIC MACROCYCLIC DERIVATIVES AS PROTEIN KINASE INHIBITORS KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2020-04-30 WO disclosed