SCHEMBL21884477

SCHEMBL21884477

Cc1ccc(O)c(C(=O)NC(=N)NCC(C)(C)O)c1-c1cccc(F)c1C

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PPIA P62937 4/20 0.36
CYP2C9 P11712 1/20 0.34
MAPK14 Q16539 1/20 0.34
CTSA P10619 1/20 0.33
NR3C1 P04150 1/20 0.32
PSMB8 P28062 1/20 0.32
PSMB5 P28074 1/20 0.32
CHRM1 P11229 2/20 0.31
BDKRB1 P46663 1/20 0.30
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21884541 0.78 PPIA (0.33) PPIA
SCHEMBL21884384 0.78 AR (0.34) PPIACHRM1
SCHEMBL21884633 0.67 CCNT1 (0.39) NR3C1
SCHEMBL15402236 0.63 CFTR (0.43) CYP2C9NR3C1CHRM1
SCHEMBL21884538 0.63 PPIA (0.35) PPIABDKRB1ADORA1
SCHEMBL21884497 0.63 PPIA (0.35) PPIA
SCHEMBL21884467 0.62 PPIA (0.38) PPIA
SCHEMBL7449035 0.61 PDE10A (0.41) CYP2C9NR3C1CHRM1
SCHEMBL15402235 0.61 NPC1 (0.40) CYP2C9NR3C1CHRM1
SCHEMBL21884563 0.61 PPIA (0.37) PPIABDKRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020061473-A1 SMALL MOLECULES TARGETING MUTANT MAMMALIAN PROTEINS JNANA THERAPEUTICS, INC. (US) 2020-03-26 WO disclosed