SCHEMBL21884863

SCHEMBL21884863

COc1cc2nccc(Oc3ccc4[nH]c(C)cc4c3F)c2cc1OC(=O)N1CCN(C)CC1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 8/20 0.62
PDGFRB P09619 3/20 0.62
AXL P30530 5/20 0.50
MET P08581 4/20 0.50
EGFR P00533 3/20 0.50
SRC P12931 3/20 0.50
TGFBR1 P36897 3/20 0.50
RET P07949 2/20 0.50
KIT P10721 2/20 0.50
FLT3 P36888 2/20 0.50
PLK4 O00444 1/20 0.50
GAK O14976 1/20 0.50
EPHB6 O15197 1/20 0.50
RIPK2 O43353 1/20 0.50
ERN1 O75460 1/20 0.50
STK10 O94804 1/20 0.50
MAP4K4 O95819 1/20 0.50
CHEK2 O96017 1/20 0.50
ABL1 P00519 1/20 0.50
ERBB2 P04626 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21884876 0.92 KDR (0.62) KDRPDGFRBAXLMETEGFR
SCHEMBL21884860 0.89 KDR (0.58) KDRPDGFRBAXLMETEGFR
SCHEMBL21884825 0.89 KDR (0.58) KDRPDGFRBAXLMETEGFR
SCHEMBL30365200 0.89 KDR (0.58) KDRPDGFRBAXLMETEGFR
SCHEMBL30365337 0.89 KDR (0.58) KDRPDGFRBAXLMETEGFR
SCHEMBL21885567 0.89 KDR (0.64) KDRPDGFRBAXLMETEGFR
SCHEMBL21886104 0.88 KDR (0.58) KDRPDGFRBAXLMETEGFR
SCHEMBL21886112 0.88 KDR (0.58) KDRPDGFRBAXLMETEGFR
SCHEMBL2062767 0.88 KDR (0.69) KDRPDGFRBAXLMETEGFR
SCHEMBL21886105 0.88 KDR (0.58) KDRPDGFRBAXLMETEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020057403-A1 INDOLE DERIVATIVE AND MEDICAL APPLICATION THEREOF 北京越之康泰生物医药科技有限公司 2020-03-26 WO disclosed