SCHEMBL21886014

SCHEMBL21886014

CC1CCCC1n1c(=O)c(C(F)F)cc2cnc(NC3CCN(S(C)(=O)=O)CC3)nc21

nearest known ligand 0.80

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCNE1 P24864 20/20 0.80
CDK2 P24941 20/20 0.80
CCND1 P24385 19/20 0.80
CDK6 Q00534 19/20 0.80
CCNT1 O60563 2/20 0.71
CDK4 P11802 2/20 0.71
CDK9 P50750 2/20 0.71
CCNE2 O96020 1/20 0.71
RB1 P06400 1/20 0.71
CDK1 P06493 1/20 0.71
CCNA2 P20248 1/20 0.71
CCND3 P30281 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22259332 1.00 CCNE1 (0.80) CCNE1CDK2CCND1CDK6CCNT1
SCHEMBL30550278 0.94 CCNE1 (0.76) CCNE1CDK2CCND1CDK6CCNT1
SCHEMBL19868252 0.93 CCNE1 (0.71) CCNE1CDK2CCND1CDK6CCNT1
SCHEMBL19868333 0.91 CCNE1 (0.78) CCNE1CDK2CCND1CDK6
SCHEMBL30550290 0.90 CCNE1 (0.70) CCNE1CDK2CCND1CDK6CCNT1
SCHEMBL19863604 0.89 CCNE1 (1.00) CCNE1CDK2CCND1CDK6CCNT1
SCHEMBL22860708 0.88 CCNE1 (0.75) CCNE1CDK2CCND1CDK6CCNT1
SCHEMBL22860657 0.88 CCNE1 (0.75) CCNE1CDK2CCND1CDK6CCNT1
SCHEMBL22860659 0.88 CCNE1 (0.75) CCNE1CDK2CCND1CDK6CCNT1
SCHEMBL29508850 0.88 CCNE1 (0.75) CCNE1CDK2CCND1CDK6CCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3497103-B1 PYRIDOPYRIMDINONE CDK2/4/6 INHIBITORS PFIZER (US) 2021-05-05 EP disclosed
WO-2020065494-A1 SYNTHESIS OF PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONES PFIZER INC. (US) 2020-04-02 WO disclosed